Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1 [E24Q]'
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Human)
Université Montpellier 1

LigandChemical structure of BindingDB Monomer ID 212436BDBM212436(JMV 3002 | N-[1-[4-[(2,4-dimethoxyphenyl)methyl]-5...)
Affinity DataKi:  8.70nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2017
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Human)
Université Montpellier 1

LigandChemical structure of BindingDB Monomer ID 50049478BDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)
Affinity DataKi:  8.90nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Human)
Université Montpellier 1

LigandChemical structure of BindingDB Monomer ID 50049478BDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)
Affinity DataKi:  68.9nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Human)
Université Montpellier 1

LigandChemical structure of BindingDB Monomer ID 212438BDBM212438(Substance P [DArg1, DTrp5,7,9, Leu11] | SPA)
Affinity DataKi:  300nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2017
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Human)
Université Montpellier 1

LigandChemical structure of BindingDB Monomer ID 212438BDBM212438(Substance P [DArg1, DTrp5,7,9, Leu11] | SPA)
Affinity DataKi:  852nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2017
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Human)
Université Montpellier 1

LigandChemical structure of BindingDB Monomer ID 212437BDBM212437(JMV 3011)
Affinity DataKi:  915nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2017
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Human)
Université Montpellier 1

LigandChemical structure of BindingDB Monomer ID 212436BDBM212436(JMV 3002 | N-[1-[4-[(2,4-dimethoxyphenyl)methyl]-5...)
Affinity DataKi:  993nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2017
Entry Details Article
PubMed