Compile Data Set for Download or QSAR
Report error Found 2228 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1/M2/M3/M4/M5'
LigandPNGBDBM50229048(CHEMBL349844)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229049(CHEMBL351934)
Affinity DataEC50:  100nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229050(CHEMBL422710)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229054(CHEMBL161748)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229057(CHEMBL161419)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229059(CHEMBL159708)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229053(CHEMBL161364)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229052(CHEMBL159651)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229051(CHEMBL159935)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229064(CHEMBL159839)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229055(CHEMBL161670)
Affinity DataEC50:  1.46E+3nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50046728(1-Methyl-5-(3-methyl-[1,2,4]oxadiazol-5-yl)-1,2,3,...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229058(CHEMBL161088)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228565(CHEMBL108557)
Affinity DataKd:  7.00E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228566(CHEMBL2092932)
Affinity DataKd:  3.23E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228567(CHEMBL2092931)
Affinity DataKd:  7.85E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228568(CHEMBL322126)
Affinity DataKd:  1.60E+4nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228569(CHEMBL1788225)
Affinity DataKd:  161nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228570(CHEMBL1788202)
Affinity DataKd:  200nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228571(CHEMBL107456)
Affinity DataKd:  97nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228572(CHEMBL432629)
Affinity DataKd:  110nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228573(CHEMBL106056)
Affinity DataKd:  3.55E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228071(CHEMBL110892)
Affinity DataKd:  1.40E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228574(CHEMBL108582)
Affinity DataKd:  8.30E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228087(CHEMBL323032)
Affinity DataKd:  1.25E+5nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228575(CHEMBL108140)
Affinity DataEC50:  2.80E+3nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228576(CHEMBL2092930)
Affinity DataKd:  80nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228577(CHEMBL1788224)
Affinity DataKd:  1.16E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataEC50:  100nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228578(CHEMBL111327)
Affinity DataKd:  4.95E+4nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228579(CHEMBL1788219)
Affinity DataKd:  6.32E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228578(CHEMBL111327)
Affinity DataEC50:  7.50E+3nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228570(CHEMBL1788202)
Affinity DataEC50:  94nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKd:  0.900nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229065(CHEMBL262517)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229067(CHEMBL355824)
Affinity DataEC50:  320nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229047(CHEMBL159628)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227302(CHEMBL154455)
Affinity DataKd:  570nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50004734(CHEMBL310852 | N-Methyl-N-(1-methyl-4-pyrrolidin-1...)
Affinity DataKd:  240nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227303(CHEMBL154092)
Affinity DataKd:  3.10E+3nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227304(CHEMBL346662)
Affinity DataKd:  5.40E+3nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227305(CHEMBL157439)
Affinity DataKd:  9.54E+4nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227306(CHEMBL346737)
Affinity DataKd:  5.00E+3nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227307(CHEMBL154320)
Affinity DataKd:  6.80E+4nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227308(CHEMBL346237)
Affinity DataKd:  8.20E+3nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227309(CHEMBL152594)
Affinity DataKd:  1.79E+4nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227310(CHEMBL155263)
Affinity DataKd:  1.30E+4nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227311(CHEMBL157438)
Affinity DataKd:  9.19E+4nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50227320(CHEMBL154627)
Affinity DataKd:  1.60E+3nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009300(CHEMBL11081 | N-Methyl-N-(4-pyrrolidin-1-yl-but-2-...)
Affinity DataKd:  2.20E+3nMAssay Description:Equilibrium dissociation constant muscarinic receptor complex, measured in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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