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Report error Found 178 Enz. Inhib. hit(s) with Target = 'Pituitary adenylate cyclase-activating polypeptide type I receptor'
LigandPNGBDBM50110068(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataKi:  56nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50122102(3-Cyano-4-hydroxy-benzoic acid [1-(2,3,5,6-tetrame...)
Affinity DataKi:  72nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374178(CHEMBL411120)
Affinity DataKi:  85nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374184(CHEMBL270677)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374179(CHEMBL409325)
Affinity DataKi:  152nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374188(CHEMBL270226)
Affinity DataKi:  167nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374187(CHEMBL256379)
Affinity DataKi:  185nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374177(CHEMBL409729)
Affinity DataKi:  204nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374180(CHEMBL404071)
Affinity DataKi:  241nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374186(CHEMBL272122)
Affinity DataKi:  274nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374183(CHEMBL269990)
Affinity DataKi:  404nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374182(CHEMBL272118)
Affinity DataKi:  522nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374181(CHEMBL256837)
Affinity DataKi:  537nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374185(CHEMBL255824)
Affinity DataKi:  554nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50110055(3-Chloro-4-hydroxy-benzoic acid [1-(4-isopropyl-be...)
Affinity DataKi:  604nMAssay Description:Displacement of [125I]PACAP27 from PAC1R expressed in HEK293f cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50550811(CHEMBL4740931)
Affinity DataIC50: <0.0100nMAssay Description:Antagonist activity at PAC1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of PACAP-induced inhibition of CREB phosphorylati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50596676(CHEMBL5203375)
Affinity DataIC50:  0.110nMAssay Description:Antagonist activity at PAC-1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of PACAP-induced increase in intracellular cAMP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50550810(CHEMBL4757203)
Affinity DataIC50:  0.182nMAssay Description:Antagonist activity at PAC1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of PACAP-induced inhibition of CREB phosphorylati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50596675(CHEMBL5208587)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at PAC-1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of PACAP-induced increase in intracellular cAMP ...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50200209(CHEMBL219499)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]PACAP27 from human PAC1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50606528(CHEMBL5219662)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity at PAC1R in human SH-SY5Y cells assessed as inhibition of PACAP38-induced cAMP accumulation pre-incubated for 30 mins followed by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50250033(CHEMBL525419 | [Ala7]PACAP38)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250074(CHEMBL507480 | [Bip6]PACAP27)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250018(CHEMBL524852 | PACAP27)
Affinity DataIC50:  4.60nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human PAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250034(CHEMBL499781 | [D-His1]PACAP27)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250077(CHEMBL503123 | [Nal6]PACAP38)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250022(CHEMBL525392 | [Ala2]PACAP27)
Affinity DataIC50:  5.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250035(CHEMBL525073 | [D-His1]PACAP38)
Affinity DataIC50:  5.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250075(CHEMBL526315 | [Bip6]PACAP38)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250059(Ac-PACAP38 | CHEMBL530563)
Affinity DataIC50:  5.70nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250019(CHEMBL524658 | PACAP | PACAP(1-38) | PACAP-38 | PA...)
Affinity DataIC50:  6.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250076(CHEMBL525613 | [Nal6]PACAP27)
Affinity DataIC50:  6.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250071(CHEMBL524683 | [Cha6]PACAP38)
Affinity DataIC50:  6.60nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250037(CHEMBL524894 | [D-Ser2]PACAP38)
Affinity DataIC50:  6.60nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250073(CHEMBL526360 | [Tyr6]PACAP38)
Affinity DataIC50:  6.70nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250069(CHEMBL524494 | [Glu3]PACAP38)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250085(CHEMBL506517 | [Aib2]PACAP38)
Affinity DataIC50:  7.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250039(CHEMBL524334 | [D-Asp3]PACAP38)
Affinity DataIC50:  7.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250036(CHEMBL506133 | [D-Ser2]PACAP27)
Affinity DataIC50:  7.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250061(CHEMBL498948 | [His(1-Me)1]PACAP38)
Affinity DataIC50:  7.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250078(CHEMBL524672 | [Pro2]PACAP27)
Affinity DataIC50:  7.80nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250072(CHEMBL498867 | [Tyr6]PACAP27)
Affinity DataIC50:  7.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250023(CHEMBL500280 | [Ala2]PACAP(1-38) | [Ala2]PACAP38)
Affinity DataIC50:  7.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250058(Ac-PACAP27 | CHEMBL505046)
Affinity DataIC50:  8.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250018(CHEMBL524852 | PACAP27)
Affinity DataIC50:  8.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250079(CHEMBL506840 | [Pro2]PACAP38)
Affinity DataIC50:  8.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250080(CHEMBL524495 | [Hyp2]PACAP27)
Affinity DataIC50:  8.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250081(CHEMBL499507 | [Hyp2]PACAP38)
Affinity DataIC50:  8.60nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250047(CHEMBL525591 | [N-Me-Ser2]PACAP38)
Affinity DataIC50:  9.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50250026(CHEMBL526899 | [Ala4]PACAP27)
Affinity DataIC50:  9.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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