Report error Found 835 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 5'
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataKd: 2.70E+5nMAssay Description:Blockade of peak K+ currents against Kv1.5 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataKd: 1.77E+5nMAssay Description:Blockade of peak K+ currents against Kv1.5 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataEC50: 900nMAssay Description:Effect on blockade of Kv1.5 channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Effect on blockade of Kv1.5 channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Effect on blockade of Kv1.5 channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataEC50: >1.10E+4nMAssay Description:Inhibition of human Kv1.5 by IonWorks patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of Kv1.5 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial myocytes by voltage-patch clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial myocytes by voltage-patch clamp electrophysiology methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human Kv1.5 expressed in mouse L929 cells assessed as inhibition of currentMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human Kv1.5 expressed in mouse L929 cells assessed as inhibition of currentMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of Kv1.5 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human Kv1.5 expressed in mouse L929 cells assessed as inhibition of currentMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of Kv1.5 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of Kv1.5 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human Kv1.5 channel expressed in CHO cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Kv1.5 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of Kv1.5 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human Kv1.5 expressed in mouse L929 cells assessed as inhibition of delayed rectifier repolarization current by patch clamp as...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human Kv1.5 transfected in mouse LTK cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of Kv1.5 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of human Kv1.5 expressed in mouse L929 cells assessed as inhibition of currentMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells assessed as blockade of ultra rapidly activating potassium current by voltage clamp t...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant human Kv1.5 expressed in mouse L929 cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Antagonist activity at human Kv1.5 expressed in mouse L929 cells assessed as inhibition of delayed rectifier repolarization current by patch clamp as...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells assessed as blockade of ultra rapidly activating potassium current by voltage clamp t...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human Kv1.5 transfected in mouse LTK cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human Kv1.5 transfected in mouse LTK cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of human KV1.5 expressed in mouse L929 cells assessed as decrease in ultrarapid potassium current amplitudeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of Kv1.5 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Kiel
Curated by ChEMBL
University of Kiel
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human Kv1.5 expressed in mouse L929 cells assessed as inhibition of delayed rectifier repolarization current by patch clamp as...More data for this Ligand-Target Pair
