Report error Found 754 Enz. Inhib. hit(s) with Target = 'Potassium-transporting ATPase alpha chain 1'
Affinity DataIC50: 4.20nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by dibutyryl cyclic adenosine 3', 5...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 36nMpH: 7.0Assay Description:Inhibition of K+ -stimulated gastric ATPase activity was measured using lyophilized gastric vesicles at pH 7More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by dibutyryl cyclic adenosine 3', 5...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by dibutyryl cyclic adenosine 3', 5...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 61nMpH: 7.0Assay Description:Inhibition of K+ -stimulated gastric ATPase activity was measured using lyophilized gastric vesicles at pH 7More data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Rat)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of rat isolated gastric (H(+)/K(+))-ATPase.More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of H+/K+ ATPase as reduced acid formation in rabbit gastric glandsMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of H+/K+ ATPase as reduced acid formation in rabbit gastric glandsMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 71nMpH: 7.0Assay Description:Inhibition of K+ -stimulated gastric ATPase activity was measured using lyophilized gastric vesicles at pH 7More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by dibutyryl cyclic adenosine 3', 5...More data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Human)
Ortho Pharmaceutical
Curated by ChEMBL
Ortho Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 92nMpH: 7.4Assay Description:Inhibition of purified H+/K+ ATPase at pH 7.4 as released inorganic phosphate from ATP using hog stomach gastric membrane vesiclesMore data for this Ligand-Target Pair
