Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3'
LigandPNGBDBM50280454((10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-3...)
Affinity DataIC50: 150nMAssay Description:Binding to PKC in 3[H]-PBDU assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2018
Entry Details

LigandPNGBDBM50368315(PROSTRATIN)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]PDBu binding to Protein kinase C of CEM cells with 10% fetal calf serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2019
Entry Details Article
PubMed
LigandPNGBDBM50281846((2R,3R)-2-Hydroxymethyl-5-oxo-4-tridec-(E)-ylidene...)
Affinity DataKi:  200nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50368315(PROSTRATIN)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]PDBu from Protein kinase C of CEM cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2019
Entry Details Article
PubMed
LigandPNGBDBM50212475(CHEMBL143453)
Affinity DataIC50: 400nMAssay Description:Binding to PKC in 3[H]-PBDU assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2018
Entry Details

LigandPNGBDBM50281845((2R,3R)-2-Hydroxymethyl-5-oxo-4-tridec-(E)-ylidene...)
Affinity DataKi:  600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50041403((2R,3R,4R)-2-Hydroxymethyl-5-oxo-4-tetradecyl-tetr...)
Affinity DataKi:  600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article