Compile Data Set for Download or QSAR
Found 5830 Enz. Inhib. hit(s) with Target = 'Receptor-type tyrosine-protein kinase FLT3 [K633Q]'
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568686(CHEMBL4864449)
Affinity DataKi:  0.100nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568690(CHEMBL4870188)
Affinity DataKi:  0.100nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355491(CHEMBL1835870)
Affinity DataKi:  0.170nMAssay Description:Inhibition of human recombinant FLT3 by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568703(CHEMBL4878159)
Affinity DataKi:  0.200nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568703(CHEMBL4878159)
Affinity DataKi: <0.300nMAssay Description:Inhibition of FLT3 D835Y mutant (unknown origin) incubated for 120 mins by ADP-glo based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568703(CHEMBL4878159)
Affinity DataKi: <0.300nMAssay Description:Inhibition of FLT3 R595_E596insEY mutant (unknown origin) incubated for 120 mins by ADP-glo based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568703(CHEMBL4878159)
Affinity DataKi: <0.300nMAssay Description:Inhibition of FLT3 F594_R595insR mutant (unknown origin) incubated for 120 mins by ADP-glo based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50020310(CHEMBL3288854)
Affinity DataKi: <0.300nMAssay Description:Binding affinity to FLT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568690(CHEMBL4870188)
Affinity DataKi:  0.400nMAssay Description:Inhibition of wild type FLT3 (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568698(CHEMBL4855435)
Affinity DataKi:  0.400nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568704(CHEMBL4867869)
Affinity DataKi:  0.600nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568691(CHEMBL4871011)
Affinity DataKi:  0.700nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568686(CHEMBL4864449)
Affinity DataKi:  0.800nMAssay Description:Inhibition of wild type FLT3 (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568691(CHEMBL4871011)
Affinity DataKi:  1nMAssay Description:Inhibition of wild type FLT3 (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355479(CHEMBL1835746)
Affinity DataKi:  1nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568704(CHEMBL4867869)
Affinity DataKi:  1nMAssay Description:Inhibition of wild type FLT3 (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568700(CHEMBL4856641)
Affinity DataKi:  2nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568687(CHEMBL4876697)
Affinity DataKi:  2nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568688(CHEMBL4862206)
Affinity DataKi:  2nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM144315(Gilteritinib | US11512074, Example T-9 | US8969336...)
Affinity DataKi:  2nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355491(CHEMBL1835870)
Affinity DataKi:  2nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50526216(CHEMBL4553725)
Affinity DataKi:  2nMAssay Description:Irreversible inhibition of recombinant human FLT3 D835Y mutant (571 to 993 residues) expressed in baculovirus expression system preincubated for 5 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355489(CHEMBL1835867)
Affinity DataKi:  2nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355464(CHEMBL1835740)
Affinity DataKi:  2.80nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568692(CHEMBL4862054)
Affinity DataKi:  4nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568688(CHEMBL4862206)
Affinity DataKi:  4nMAssay Description:Inhibition of wild type FLT3 (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568698(CHEMBL4855435)
Affinity DataKi:  4nMAssay Description:Inhibition of wild type FLT3 (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355480(CHEMBL1835747)
Affinity DataKi:  5nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355490(CHEMBL1835869)
Affinity DataKi:  5nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355482(CHEMBL1835749)
Affinity DataKi:  5nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355492(CHEMBL1835871)
Affinity DataKi:  5nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50341530(3-(4-(Piperidin-1-yl)benzoylamino)-5-(2-(methylami...)
Affinity DataKi:  5nMAssay Description:Inhibition of FMSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50277622(CHEMBL4162390)
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant human FLT3 using EAIYAAPFAKKK as substrate by ATP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50341521(3-(4-(Piperidin-1-yl)benzoylamino)-5-(2-(methylami...)
Affinity DataKi:  6nMAssay Description:Inhibition of FMSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355467(CHEMBL1833992)
Affinity DataKi:  6nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355483(CHEMBL1835750)
Affinity DataKi:  7nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568699(CHEMBL4866028)
Affinity DataKi:  7nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50277601(CHEMBL4167646)
Affinity DataKi:  7nMAssay Description:Inhibition of recombinant human FLT3 using EAIYAAPFAKKK as substrate by ATP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50341542(3-(4-Dimethylaminobenzoylamino)-5-(pyridin-4-yl)-(...)
Affinity DataKi:  8nMAssay Description:Inhibition of FMSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355481(CHEMBL1835748)
Affinity DataKi:  8nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355488(CHEMBL1835866)
Affinity DataKi:  9nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568687(CHEMBL4876697)
Affinity DataKi:  9nMAssay Description:Inhibition of wild type FLT3 (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355486(CHEMBL1835864)
Affinity DataKi:  10nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM144315(Gilteritinib | US11512074, Example T-9 | US8969336...)
Affinity DataKi:  10nMAssay Description:Inhibition of wild type FLT3 (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50526217(CHEMBL4442997)
Affinity DataKi:  10nMAssay Description:Irreversible inhibition of recombinant human FLT3 D835Y mutant (571 to 993 residues) expressed in baculovirus expression system preincubated for 5 to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50341540(3-(4-tert-Butylbenzoylamino)-5-(pyridin-4-yl)-(1H)...)
Affinity DataKi:  11nMAssay Description:Inhibition of FMSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50568695(CHEMBL4865261)
Affinity DataKi:  11nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) using Glu/Tyr peptide substrate incubated for 120 mins measured after 40 mins incubation under dark by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355493(CHEMBL1835736)
Affinity DataKi:  11nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355485(CHEMBL1835863)
Affinity DataKi:  11nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3 [K633Q](Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50355468(CHEMBL1835743)
Affinity DataKi:  12nMAssay Description:Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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