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Report error Found 14 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor alpha [200-419]'
TargetRetinoic acid receptor alpha [200-419]/gamma [183-417](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36811(BMS614)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419]/gamma [183-417](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36810(BMS753 | US9963439, BMS753)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36810(BMS753 | US9963439, BMS753)
Affinity DataKi:  2nM ΔG°:  -46.2kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36811(BMS614)
Affinity DataKi:  2.5nM ΔG°:  -45.6kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31887(BMS181156 | Ch 80)
Affinity DataKd:  0.400nMpH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31888(CD666)
Affinity DataKd:  2.24E+3nMpH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31890(BMS270395)
Affinity DatapH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKd:  0.400nMpH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKd:  0.300nMpH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31886(CD564 | CHEMBL309282)
Affinity DataKd:  118nMpH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31885(BMS184394 | CHEMBL82089)
Affinity DataKd:  7.50E+3nMpH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31884(BMS184394-S | CHEMBL81273)
Affinity DataKd:  7.50E+3nMpH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31882(BMS184394-R | CHEMBL80992)
Affinity DataKd:  1.60E+4nMpH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31889(BMS 961 | BMS270394 | BMS961)
Affinity DatapH: 7.9 T: 4°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed