Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with Target = 'Sensory histidine kinase DcuS'
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497020(CHEMBL3235590)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataEC50:  26nMAssay Description:Effective concentration to antagonise accessory gene regulator C3 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151882([15-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataEC50:  1.10E+4nMAssay Description:Effective concentration to antagonise accessory gene regulator C1 of Staphylococcus aureus; range = 9-11 uMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(GVNACSSLF | CHEMBL182783)
Affinity DataEC50:  3.60nMAssay Description:Effective concentration to antagonise accessory gene regulator C2 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(YSTCYFIM | CHEMBL426697)
Affinity DataEC50:  13nMAssay Description:Effective concentration to antagonise accessory gene regulator C4 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497017(CHEMBL3235596)
Affinity DataKd:  2.30E+4nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497018(CHEMBL3235589)
Affinity DataKd:  7.20E+4nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497019(CHEMBL3235588)
Affinity DataKd:  2.58E+5nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497021(CHEMBL3235597)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497022(CHEMBL1213657)
Affinity DataKd:  2.22E+5nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-Met) | CHEMBL362...)
Affinity DataIC50: 0.300nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 0.300nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(GVNACSSLF | CHEMBL182783)
Affinity DataIC50: 1nMAssay Description:Concentration required to antagonise accessory gene regulator C3 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50526860(CHEMBL4554516)
Affinity DataIC50: 1nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(YSTCYFIM | CHEMBL426697)
Affinity DataIC50: 1nMAssay Description:Concentration required to antagonise accessory gene regulator C3 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151873(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 2.80nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(GVNACSSLF | CHEMBL182783)
Affinity DataIC50: 2.90nMAssay Description:Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50020375(CHEMBL3289785)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50526861(CHEMBL2337554)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN8463 assessed as beta-lactamase activity incubated for 80 mins by spectrophotomet...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50020375(CHEMBL3289785)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN8463 assessed as beta-lactamase activity incubated for 80 mins by spectrophotomet...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50526861(CHEMBL2337554)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus SA502A assessed as beta-lactamase activity incubated for 80 mins by spectrophotomet...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(YSTCYFIM | CHEMBL426697)
Affinity DataIC50: 4nMAssay Description:Concentration required to antagonise accessory gene regulator C2 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151877(N-[9-Benzyl-6-sec-butyl-12-methyl-3-(2-methylsulfa...)
Affinity DataIC50: 5nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151877(N-[9-Benzyl-6-sec-butyl-12-methyl-3-(2-methylsulfa...)
Affinity DataIC50: 5nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50: 6nMAssay Description:Concentration required to antagonise accessory gene regulator C2 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50526859(CHEMBL4518791)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-Met) | CHEMBL362...)
Affinity DataIC50: 8nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 10nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 10nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151883(N-[9-Benzyl-6-sec-butyl-12-methyl-3-(2-methylsulfa...)
Affinity DataIC50: 19nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-Met) | CHEMBL362...)
Affinity DataIC50: 21nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-Met) | CHEMBL362...)
Affinity DataIC50: 21nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50: 70nMAssay Description:Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(GVNACSSLF | CHEMBL182783)
Affinity DataIC50: 86nMAssay Description:Concentration required to antagonise accessory gene regulator C4 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151873(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 137nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50: 150nMAssay Description:Concentration required to antagonise accessory gene regulator C4 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 230nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151878(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 256nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151878(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 256nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151883(N-[9-Benzyl-6-sec-butyl-12-methyl-3-(2-methylsulfa...)
Affinity DataIC50: 295nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151872(2-{2-[4-(4-Benzoyl-phenoxy)-butyrylamino]-3-hydrox...)
Affinity DataIC50: 303nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151872(2-{2-[4-(4-Benzoyl-phenoxy)-butyrylamino]-3-hydrox...)
Affinity DataIC50: 303nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406396(CHEMBL4159129)
Affinity DataIC50: 456nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406468(CHEMBL4169564)
Affinity DataIC50: 608nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406354(CHEMBL4169312)
Affinity DataIC50: 622nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406399(CHEMBL4161642)
Affinity DataIC50: 738nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406469(CHEMBL4174843)
Affinity DataIC50: 913nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406360(CHEMBL4167382)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151875(N-(3-Benzyl-9,12-bis-hydroxymethyl-6-isobutyl-2,5,...)
Affinity DataIC50: 4.00E+3nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151875(N-(3-Benzyl-9,12-bis-hydroxymethyl-6-isobutyl-2,5,...)
Affinity DataIC50: 4.00E+3nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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