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Report error Found 1724 Enz. Inhib. hit(s) with Target = 'Substance-K receptor'
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476247(CHEMBL224081)
Affinity DataKi:  0.0251nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50404016(CHEMBL2112922)
Affinity DataKi:  0.0500nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415924(CHEMBL1083850)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50404016(CHEMBL2112922)
Affinity DataKi:  0.0501nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476235(CHEMBL436981)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476788(CHEMBL243711)
Affinity DataKi:  0.0525nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476771(CHEMBL244362)
Affinity DataKi:  0.0575nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476748(CHEMBL395972)
Affinity DataKi:  0.0603nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476221(CHEMBL387506)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476233(CHEMBL439281)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476750(Ibodutant | MEN-15596)
Affinity DataKi:  0.0759nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415954(CHEMBL1083858)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415966(CHEMBL1083974)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476764(CHEMBL395974)
Affinity DataKi:  0.0977nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472916(CHEMBL223221 | MEN-11690)
Affinity DataKi:  0.100nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472916(CHEMBL223221 | MEN-11690)
Affinity DataKi:  0.100nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476219(CHEMBL225297)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212987(CHEMBL2110370 | GR-159897)
Affinity DataKi:  0.100nMAssay Description:Binding affinity by displacement of radiolabeled GR-100679 from Tachykinin receptor 2 from homogenized rat colonMore data for this Ligand-Target Pair
In DepthDetails
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472916(CHEMBL223221 | MEN-11690)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415928(CHEMBL1083879)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476250(CHEMBL389510)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476754(CHEMBL242626)
Affinity DataKi:  0.117nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476229(CHEMBL224374)
Affinity DataKi:  0.126nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476251(CHEMBL224003)
Affinity DataKi:  0.126nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50404025(CHEMBL2112925)
Affinity DataKi:  0.126nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415949(CHEMBL1083863)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415943(CHEMBL1083869)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476793(CHEMBL394780)
Affinity DataKi:  0.132nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476753(CHEMBL395973)
Affinity DataKi:  0.141nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50469874(CHEMBL59780)
Affinity DataKi:  0.155nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50048413(CHEMBL2370064)
Affinity DataKi:  0.155nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415970(CHEMBL1083870)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415940(CHEMBL1083873)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415939(CHEMBL1083874)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50415938(CHEMBL1083875)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476244(CHEMBL389511)
Affinity DataKi:  0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473829(CHEMBL389459 | MEN-11995)
Affinity DataKi:  0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476223(CHEMBL413715)
Affinity DataKi:  0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476222(CHEMBL266284)
Affinity DataKi:  0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473829(CHEMBL389459 | MEN-11995)
Affinity DataKi:  0.158nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476231(CHEMBL225588)
Affinity DataKi:  0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476220(CHEMBL225392)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476256(CHEMBL388626)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476253(CHEMBL389279)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476236(CHEMBL224009)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50116083(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50116745(CHEMBL78284 | N-{(R)-5-[4-(3-Carbamoylmethyl-2-oxo...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against recombinant human tachykinin receptor 2 in CHO cells using [3H]-NKA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50476766(CHEMBL243496)
Affinity DataKi:  0.224nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50418024(CHEMBL1683146)
Affinity DataKi:  0.234nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 1724 total ) | Next | Last >>
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