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Report error Found 9 Enz. Inhib. hit(s) with Target = 'Sulfotransferase 2A1'
TargetSulfotransferase 2A1(Human)
Albert Einstein College of Medicine

LigandPNGBDBM50176062(3-(5H-dibenzo[a,d][7]annulen-5-yl)-N-methylpropan-...)
Affinity DataKi:  7.60E+4nM ΔG°:  -21.7kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 2A1(Human)
Albert Einstein College of Medicine

LigandPNGBDBM22870(13-chloro-10-(piperazin-1-yl)-2-oxa-9-azatricyclo[...)
Affinity DataKi:  1.25E+5nM ΔG°:  -20.6kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 2A1(Human)
Albert Einstein College of Medicine

LigandPNGBDBM50380592(CHEMBL1552719)
Affinity DataIC50:  50nMAssay Description:Affinity for CCK2 receptor assessed by inhibition of pentagastrin-stimulated acid secretion in perfused rat stomachMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Human)
Albert Einstein College of Medicine

LigandPNGBDBM50427989(CHEMBL2325503)
Affinity DataIC50:  1.01E+3nMAssay Description:Affinity for CCK2 receptor assessed by inhibition of pentagastrin-stimulated acid secretion in perfused rat stomachMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Rat)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Rat)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Rat)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM7462(3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Rat)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM23420(7,4′-Dihydroxy-isoflavone (3a) | 7-hydroxy-3...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50051828(2-(4-hydroxyphenyl)-3-methyl-1-(2,3,4,5,6-pentaflu...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibitory activity against dehydroepiandrosterone sulfatase (DHA-STS)More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed