Compile Data Set for Download or QSAR
Report error Found 1046 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 3'
LigandPNGBDBM776072((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 2.01nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776069((S)-(5-(2-ethylphenoxy)-2-(3-(3-methylpyridin-2-yl...)
Affinity DataIC50: 2.54nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776067((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 2.65nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776069((S)-(5-(2-ethylphenoxy)-2-(3-(3-methylpyridin-2-yl...)
Affinity DataIC50: 2.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776019((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 3.91nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776197((3-(2'-cyclopropyl-3-(hydroxymethyl)biphenyl-4-yl)...)
Affinity DataIC50: 3.99nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776185((5-fluoropyridin-2-yl)(3-(3-(hydroxymethyl)-2'-iso...)
Affinity DataIC50: 5.56nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776071((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 7.44nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776122(US12435061, Compound 1-316)
Affinity DataIC50: 7.77nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776033(US12435061, Compound 1-236)
Affinity DataIC50: 8.27nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776047((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 8.42nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776071((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 9.39nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776224(US12435061, Compound KM-085)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775687(US12435061, Compound 2-67.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776219(US12435061, Compound KM-054-E1)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775697(US12435061, Compound 2-72.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775666(US12435061, Compound 2-53.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776208(US12435061, Compound KM-001-E1)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775664(US12435061, Compound 2-51.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775716(US12435061, Compound 2-77.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775625(US12435061, Compound 2-30.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775624(US12435061, Compound 2-29.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775671(US12435061, Compound 2-57.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776213(US12435061, Compound KM-023-E1)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775670(US12435061, Compound 2-56.)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776211(US12435061, Compound KM-002-E1)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776210(US12435061, Compound KM-002)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775943((S)-(2'-ethyl-4-(3-(5-(trifluoromethyl)pyridin-2-y...)
Affinity DataIC50: 10.7nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776128(US12435061, Compound 1-321)
Affinity DataIC50: 12.2nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776045((S)-(5-(3-chlorophenoxy)-2-(3-(3-chloropyridin-2-y...)
Affinity DataIC50: 12.3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776066((S)-(2-(3-(3-chloropyridin-2-ylamino)pyrrolidin-1-...)
Affinity DataIC50: 12.6nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776020((S)-(5-(2-chlorophenoxy)-2-(3-(3-chloropyridin-2-y...)
Affinity DataIC50: 13.3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776134((S)-2-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-...)
Affinity DataIC50: 15.9nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776038((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 18.6nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776068((S)-(5-(2-ethylphenoxy)-2-(3-(3-fluoropyridin-2-yl...)
Affinity DataIC50: 19.1nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776032(US12435061, Compound 1-235)
Affinity DataIC50: 19.9nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775946((S)-(2'-(trifluoromethyl)-4-(3-(5-(trifluoromethyl...)
Affinity DataIC50: 20.4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776123(US12435061, Compound 1-317)
Affinity DataIC50: 20.8nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776030((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 21.6nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776046((S)-(5-(4-chlorophenoxy)-2-(3-(3-chloropyridin-2-y...)
Affinity DataIC50: 22.1nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776057((S)-(2-(3-(3-chloropyridin-2-ylamino)pyrrolidin-1-...)
Affinity DataIC50: 23.3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775933((S)-(6-phenoxy-3-(3-(5-(trifluoromethyl)pyridin-2-...)
Affinity DataIC50: 23.6nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776061((2-chlorophenyl)(4-((S)-3-(3-chloropyridin-2-yloxy...)
Affinity DataIC50: 23.7nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776076(US12435061, Compound 1-275)
Affinity DataIC50: 24.8nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776048((S)-(2-(3-(3-chloropyridin-2-ylamino)pyrrolidin-1-...)
Affinity DataIC50: 25.6nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776175((5-fluoropyridin-2-yl)(3-(2-(hydroxymethyl)-4-(2-i...)
Affinity DataIC50: 25.7nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776163(US12435061, Compound 1-353)
Affinity DataIC50: 26.8nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776140((S)-2-(2-(3-(3-fluoropyridin-2-yloxy)pyrrolidin-1-...)
Affinity DataIC50: 28nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM775969((S)-(2-(3-(3-chloropyridin-2-yloxy)pyrrolidin-1-yl...)
Affinity DataIC50: 29nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

LigandPNGBDBM776065((S)-(5-(2-chlorophenoxy)-2-(3-(3-chloropyridin-2-y...)
Affinity DataIC50: 30.9nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent

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