Compile Data Set for Download or QSAR
Report error Found 542 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor'
LigandChemical structure of BindingDB Monomer ID 50030815BDBM50030815(CHEMBL404594)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469937BDBM50469937(CHEMBL104493)
Affinity DataKi:  0.126nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50230790BDBM50230790(CHEMBL292892)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50230779BDBM50230779(CHEMBL294686)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469896BDBM50469896(CHEMBL326910)
Affinity DataKi:  0.316nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50030815BDBM50030815(CHEMBL404594)
Affinity DataIC50: 0.350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469939BDBM50469939(CHEMBL323125)
Affinity DataKi:  0.398nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469890BDBM50469890(CHEMBL63072)
Affinity DataKi:  0.398nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50230811BDBM50230811(CHEMBL293091)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228201BDBM50228201(CHEMBL265084)
Affinity DataKi:  0.460nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469901BDBM50469901(SAPRISARTAN | GR-138950)
Affinity DataKi:  0.501nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50230778BDBM50230778(CHEMBL56211)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50230771BDBM50230771(CHEMBL55510)
Affinity DataIC50: 0.590nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469888BDBM50469888(CHEMBL104667)
Affinity DataKi:  0.631nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228201BDBM50228201(CHEMBL265084)
Affinity DataKi:  0.740nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469892BDBM50469892(CHEMBL107081)
Affinity DataKi:  0.794nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469886BDBM50469886(CHEMBL107006)
Affinity DataKi:  0.794nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50230806BDBM50230806(CHEMBL294415)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228204BDBM50228204(CHEMBL405389)
Affinity DataKi:  0.850nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469893BDBM50469893(CHEMBL104418)
Affinity DataKi:  1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469940BDBM50469940(CHEMBL105887)
Affinity DataKi:  1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50048078BDBM50048078(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228203BDBM50228203(CHEMBL262025)
Affinity DataKi:  1nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469897BDBM50469897(CHEMBL104281)
Affinity DataKi:  1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228204BDBM50228204(CHEMBL405389)
Affinity DataKi:  1.20nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50212829BDBM50212829(CHEMBL170944)
Affinity DataIC50: 1.20nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50469938BDBM50469938(CHEMBL322989)
Affinity DataKi:  1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469889BDBM50469889(CHEMBL62553)
Affinity DataKi:  1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469934BDBM50469934(CHEMBL324196)
Affinity DataKi:  1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469935BDBM50469935(CHEMBL62909)
Affinity DataKi:  1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50042235BDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50228195BDBM50228195(CHEBI:2719 | Angiotensin Ii)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50236697BDBM50236697(L-alpha-aspartyl-L-arginyl-L-valyl-L-tyrosyl-L-iso...)
Affinity DataKi:  1.40nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228198BDBM50228198(CHEMBL414796)
Affinity DataKi:  1.5nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50011975BDBM50011975(4-[2-Butyl-5-(2-carboxy-3-thiophen-2-yl-propenyl)-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228894BDBM50228894(CHEMBL312754)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228199BDBM50228199(Angiotensinamide | ANGIOTENSIN AMIDE)
Affinity DataKi:  1.60nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469887BDBM50469887(CHEMBL107043)
Affinity DataKi:  1.60nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469899BDBM50469899(CHEMBL107967)
Affinity DataKi:  1.60nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228200BDBM50228200(CHEMBL217516)
Affinity DataKi:  1.60nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228203BDBM50228203(CHEMBL262025)
Affinity DataKi:  1.70nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50228198BDBM50228198(CHEMBL414796)
Affinity DataKi:  1.80nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50236697BDBM50236697(L-alpha-aspartyl-L-arginyl-L-valyl-L-tyrosyl-L-iso...)
Affinity DataKi:  1.90nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469891BDBM50469891(CHEMBL322516)
Affinity DataKi:  2nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50469900BDBM50469900(CHEMBL104252)
Affinity DataKi:  2nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50236697BDBM50236697(L-alpha-aspartyl-L-arginyl-L-valyl-L-tyrosyl-L-iso...)
Affinity DataIC50: 2nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50212650BDBM50212650(CHEMBL89917)
Affinity DataKi:  2.10nMAssay Description:Tested for binding affinity by measuring displacement of [125I]-Sar1 Ile8 angiotensin II from rat adrenal cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50281848BDBM50281848(L-158827 | 2-Ethyl-5,7-dimethyl-3-{4-[2-(2H-tetraz...)
Affinity DataIC50: 2.30nMAssay Description:Compound was tested for inhibition of Angiotensin II receptor in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50212853BDBM50212853(CHEMBL274626)
Affinity DataIC50: 2.40nMAssay Description:Compound was tested for inhibition of Angiotensin II receptor in rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50469894BDBM50469894(CHEMBL323315)
Affinity DataKi:  2.5nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
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