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Report error Found 1251 Enz. Inhib. hit(s) with Target = 'Vasopressin V1b receptor'
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50345133((S)-1-((R)-5-chloro-3-(2-methoxy-5-(pyrrolidin-1-y...)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50345134((S)-1-((R)-5-chloro-3-(2-methoxy-5-((4-methylpiper...)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205313(CHEMBL265859 | d[Leu4]AVP)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50345131((S)-1-((R)-5-chloro-3-(2-methoxy-4-((4-methylpiper...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50345130((S)-1-((R)-5-chloro-3-(2-methoxy-4-(pyrrolidin-1-y...)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205305(CHEMBL375324 | d[Arg4]AVP)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205309(CHEMBL412972 | d[Leu4,Lys8]VP)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205296(CHEMBL385739 | d[Arg4,Dab8]VP)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145126((2S)-2-{[(2R)-1-{[(4S,7R,10S,13R,16S)-13-benzyl-7-...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205300(CHEMBL221436 | d[Val4]AVP)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205297(CHEMBL412973 | d[Leu4,Dab8]VP)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50345132((S)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulfonyl...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205301(CHEMBL375188 | d[Leu4,Orn8]VP)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145118(CHEMBL412353 | d[Val4]AVP)
Affinity DataKi:  0.290nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145112((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205303(CHEMBL373968 | d[Leu4,Dap8]VP)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50370387(CHEMBL1790575)
Affinity DataKi:  0.420nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145124((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-10-but...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205311(CHEMBL375096 | d[Orn4]AVP)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205306(CHEMBL375323 | d[Orn4,Lys8]VP)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145107((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-10-(3-aminopropy...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]-AVP from human vasopressin V1b receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145117((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50342028(2-((S)-6-amino-2-((S)-1-((4R,7S,10S,13S,16S)-7-(2-...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.590nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205292(CHEMBL385068 | d[Arg4,Orn8]VP)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205298(CHEMBL375325 | d[Arg4,Lys8]VP)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50299343((2S,4R)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulf...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]Arg8-vasopressin from human vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50299343((2S,4R)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulf...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50342032(2-((S)-2-((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-...)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50342029(2-((S)-2-((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50145108((2S)-2-{[(2R)-1-{[(4S,7R,13R,16S)-13-benzyl-7-(car...)
Affinity DataKi:  0.780nMAssay Description:Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT recepto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205307(CHEMBL412742 | d[Cha4,Dab8]VP)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50345129((S)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulfonyl...)
Affinity DataKi:  0.810nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205310(CHEMBL219272 | d[Orn4,Orn8]VP)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175037(US9688678, 9A (+)-3-(2-ethoxy-3-pyridyl)-1-[(5-met...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM174904(US9688678, 1A (+)-3-(2-ethoxy-5-methoxy-phenyl)-1-...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175039(US9688678, 11 (+)-3-(2-ethoxy-5-methoxyphenyl)-1-(...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299343((2S,4R)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulf...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]Arg8-vasopressin from rat vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175212(US9688678, 34 (3S)-1-[(5-chloro-2-pyridyl)sulfonyl...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175064(US9688678, 25 (+)-3-(2-ethoxy-5-methoxy-phenyl)-1-...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175060(US9688678, 21 (+-)-3-(2,5-dimethoxyphenyl)-1-[(5-m...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175058(US9688678, 19 (+-)-3-(2-ethoxy-5-methoxy-phenyl)-3...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175057(US9688678, 18A (+)-3-(2-methoxyphenyl)-1-[(5-metho...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175056(US9688678, 18 (+-)3-(2-methoxyphenyl)-1-[(5-methox...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175055(US9688678, 17B (+)-3-(2-ethoxy-5-methoxy-phenyl)-1...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM175054(US9688678, 17 (+-)-3-(2-ethoxy-5-methoxy-phenyl)-1...)
Affinity DataKi: <1nM ΔG°: <-51.4kJ/molepH: 7.4 T: 25°CAssay Description:The binding assay was carried out by the method based on that of Tahara et al. (Tahara A et al., Brit. J. Pharmacol. 125, 1463-1470 (1998)). The incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299343((2S,4R)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulf...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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