Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50035050
TargetD(1A) dopamine receptor(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  0.120nMAssay Description:Compound was evaluated for affinity towards dopamine D1-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088753(5-(3-Bromo-phenyl)-8-chloro-3-methyl-2,3,4,5-tetra...)
Affinity DataKi:  0.260nMAssay Description:Compound was evaluated for affinity towards dopamine D1-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088754(Cyclopentadienyltricarbonylrheniumbenzazepine (2`-...)
Affinity DataKi:  0.610nMAssay Description:Compound was evaluated for affinity towards dopamine D1-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088755(SCH-23390 | 5-(2-Bromo-phenyl)-8-chloro-3-methyl-2...)
Affinity DataKi:  0.700nMAssay Description:Compound was evaluated for affinity towards dopamine D1-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088753(5-(3-Bromo-phenyl)-8-chloro-3-methyl-2,3,4,5-tetra...)
Affinity DataKi:  2.80nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2C receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088756(Cyclopentadienyltricarbonylrheniumbenzazepine (3`-...)
Affinity DataKi:  2.90nMAssay Description:Compound was evaluated for affinity towards dopamine D1-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088753(5-(3-Bromo-phenyl)-8-chloro-3-methyl-2,3,4,5-tetra...)
Affinity DataKi:  8.5nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2A receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2A receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088755(SCH-23390 | 5-(2-Bromo-phenyl)-8-chloro-3-methyl-2...)
Affinity DataKi:  12nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2C receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  13nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2C receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088754(Cyclopentadienyltricarbonylrheniumbenzazepine (2`-...)
Affinity DataKi:  17nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2A receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088755(SCH-23390 | 5-(2-Bromo-phenyl)-8-chloro-3-methyl-2...)
Affinity DataKi:  22nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2A receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088754(Cyclopentadienyltricarbonylrheniumbenzazepine (2`-...)
Affinity DataKi:  29nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2C receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088756(Cyclopentadienyltricarbonylrheniumbenzazepine (3`-...)
Affinity DataKi:  106nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2C receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088756(Cyclopentadienyltricarbonylrheniumbenzazepine (3`-...)
Affinity DataKi:  227nMAssay Description:Compound was evaluated for affinity towards cerebral 5-hydroxytryptamine 2A receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Mouse)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088754(Cyclopentadienyltricarbonylrheniumbenzazepine (2`-...)
Affinity DataKi:  549nMAssay Description:Compound was evaluated for affinity towards dopamine D2-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Mouse)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088755(SCH-23390 | 5-(2-Bromo-phenyl)-8-chloro-3-methyl-2...)
Affinity DataKi:  583nMAssay Description:Compound was evaluated for affinity towards dopamine D2-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Mouse)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088753(5-(3-Bromo-phenyl)-8-chloro-3-methyl-2,3,4,5-tetra...)
Affinity DataKi:  1.12E+3nMAssay Description:Compound was evaluated for affinity towards dopamine D2-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Mouse)
Yale University

Curated by ChEMBL
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  1.21E+3nMAssay Description:Compound was evaluated for affinity towards dopamine D2-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Mouse)
Yale University

Curated by ChEMBL
LigandPNGBDBM50088756(Cyclopentadienyltricarbonylrheniumbenzazepine (3`-...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for affinity towards dopamine D2-like receptor in homogenate of caudate putamen tissue from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed