Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50011269
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104419BDBM50104419(Glutamyl-gamma-boronate analogue | CHEMBL85937)
Affinity DataIC50: 50nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104415BDBM50104415((S)-2-Amino-4-((1R,5S)-5,9,9-trimethyl-2,4-dioxa-3...)
Affinity DataIC50: 70nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104413BDBM50104413(Glutamyl-gamma-boronate analogue | CHEMBL87796)
Affinity DataIC50: 100nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104433BDBM50104433((S)-2-Methylamino-4-((1R,5S)-5,9,9-trimethyl-2,4-d...)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104419BDBM50104419(Glutamyl-gamma-boronate analogue | CHEMBL85937)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104415BDBM50104415((S)-2-Amino-4-((1R,5S)-5,9,9-trimethyl-2,4-dioxa-3...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104413BDBM50104413(Glutamyl-gamma-boronate analogue | CHEMBL87796)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104428BDBM50104428(N-[(S)-2-Amino-4-((1R,5S)-5,9,9-trimethyl-2,4-diox...)
Affinity DataIC50: 4.70E+3nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104432BDBM50104432(3-Amino-5-((1R,5S)-5,9,9-trimethyl-2,4-dioxa-3-bor...)
Affinity DataIC50: 6.50E+3nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104422BDBM50104422(4-Amino-N-[(S)-2-amino-4-((1R,5S)-5,9,9-trimethyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory concentration against transferase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104429BDBM50104429((S)-2-Acetylamino-4-((1R,5S)-5,9,9-trimethyl-2,4-d...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against transferase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104424BDBM50104424((S)-2-Amino-5-((1R,5S)-5,9,9-trimethyl-2,4-dioxa-3...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104425BDBM50104425((S)-2-Amino-5-((1R,5S)-5,9,9-trimethyl-2,4-dioxa-3...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104421BDBM50104421((S)-2-Benzyloxycarbonylamino-5-((1R,5S)-5,9,9-trim...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104430BDBM50104430((S)-2-Benzyloxycarbonylamino-5-((1R,5S)-5,9,9-trim...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104427BDBM50104427([3-((1R,5S)-5,9,9-Trimethyl-2,4-dioxa-3-bora-tricy...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104420BDBM50104420((S)-2-Amino-N-methylcarbamoylmethyl-4-((1R,5S)-5,9...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104431BDBM50104431(3-((1R,5S)-5,9,9-Trimethyl-2,4-dioxa-3-bora-tricyc...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against transferase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104426BDBM50104426((S)-2-(2-Amino-acetylamino)-4-((1R,5S)-5,9,9-trime...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104418BDBM50104418(N-[(S)-2-Amino-4-((1R,5S)-5,9,9-trimethyl-2,4-diox...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104414BDBM50104414((S)-2-Benzyloxycarbonylamino-4-((1R,5S)-5,9,9-trim...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104423BDBM50104423((S)-2-Amino-N-methyl-4-((1R,5S)-5,9,9-trimethyl-2,...)
Affinity DataIC50: 3.50E+4nMAssay Description:In vitro inhibitory concentration against transferase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104420BDBM50104420((S)-2-Amino-N-methylcarbamoylmethyl-4-((1R,5S)-5,9...)
Affinity DataIC50: 4.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104418BDBM50104418(N-[(S)-2-Amino-4-((1R,5S)-5,9,9-trimethyl-2,4-diox...)
Affinity DataIC50: 4.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104428BDBM50104428(N-[(S)-2-Amino-4-((1R,5S)-5,9,9-trimethyl-2,4-diox...)
Affinity DataIC50: 5.50E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104426BDBM50104426((S)-2-(2-Amino-acetylamino)-4-((1R,5S)-5,9,9-trime...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104429BDBM50104429((S)-2-Acetylamino-4-((1R,5S)-5,9,9-trimethyl-2,4-d...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104421BDBM50104421((S)-2-Benzyloxycarbonylamino-5-((1R,5S)-5,9,9-trim...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104424BDBM50104424((S)-2-Amino-5-((1R,5S)-5,9,9-trimethyl-2,4-dioxa-3...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104423BDBM50104423((S)-2-Amino-N-methyl-4-((1R,5S)-5,9,9-trimethyl-2,...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104422BDBM50104422(4-Amino-N-[(S)-2-amino-4-((1R,5S)-5,9,9-trimethyl-...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104430BDBM50104430((S)-2-Benzyloxycarbonylamino-5-((1R,5S)-5,9,9-trim...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104425BDBM50104425((S)-2-Amino-5-((1R,5S)-5,9,9-trimethyl-2,4-dioxa-3...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104414BDBM50104414((S)-2-Benzyloxycarbonylamino-4-((1R,5S)-5,9,9-trim...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104427BDBM50104427([3-((1R,5S)-5,9,9-Trimethyl-2,4-dioxa-3-bora-tricy...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104417BDBM50104417((S)-2-Amino-4-((1R,5S)-5,9,9-trimethyl-2,4-dioxa-3...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104416BDBM50104416((S)-2-Benzyloxycarbonylamino-4-((1R,5S)-5,9,9-trim...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamyl-tRNA(Gln) amidotransferase subunit C(Streptococcus pyogenes M1 GAS)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104431BDBM50104431(3-((1R,5S)-5,9,9-Trimethyl-2,4-dioxa-3-bora-tricyc...)
Affinity DataIC50: 8.00E+4nMAssay Description:In vitro inhibitory concentration against Glutaminase activity of bacterial Glu-tRNA-Gln aminotransferase (Glu-AdT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed