Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50011905
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50078572(CHEMBL297496 | {4-[(4-Dimethylamino-phenyl)-(4-{3-...)
Affinity DataKd:  1.20nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111931(Phosphoric acid 3-(4-pyren-1-yl-butyrylamino)-prop...)
Affinity DataKd:  140nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111931(Phosphoric acid 3-(4-pyren-1-yl-butyrylamino)-prop...)
Affinity DataKd:  140nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111928(Phosphoric acid 3-[(naphthalene-1-carbonyl)-amino]...)
Affinity DataKd:  160nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111928(Phosphoric acid 3-[(naphthalene-1-carbonyl)-amino]...)
Affinity DataKd:  160nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataKd:  260nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111932(inositol 1,4,5-Trisphosphate analogue | CHEMBL3694...)
Affinity DataKd:  620nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50078573(Phosphoric acid 3-amino-propyl ester (1R,2R,3S,4R,...)
Affinity DataKd:  1.50E+3nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111929(Phosphoric acid 3-{4-[bis-(4-dimethylamino-phenyl)...)
Affinity DataKd:  3.20E+3nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111929(Phosphoric acid 3-{4-[bis-(4-dimethylamino-phenyl)...)
Affinity DataKd:  3.20E+3nMAssay Description:Dissociation constant using IP3-binding domain (IBD) of human Type 1 inositol 1,4,5-trisphosphate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed