Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50013758
TargetCoagulation factor VII(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14597(2-[3-Amino-3-fluoro-4-(isopropylamino)-1,1-bipheny...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity of the compound against tissue coagulation factor VIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14597(2-[3-Amino-3-fluoro-4-(isopropylamino)-1,1-bipheny...)
Affinity DataIC50:  950nMAssay Description:Inhibitory activity of the compound against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14601(CHEMBL125585 | N-[(4-carbamimidoylphenyl)methyl]-2...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity of the compound against tissue coagulation factor VIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50134405(CHEMBL421098 | N-(4-Carbamimidoyl-benzyl)-2-(5-iso...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory activity of the compound against tissue coagulation factor VIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14599(CHEMBL333980 | N-[(4-carbamimidoylphenyl)methyl]-2...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibitory activity of the compound against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14599(CHEMBL333980 | N-[(4-carbamimidoylphenyl)methyl]-2...)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibitory activity of the compound against tissue coagulation factor VIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14597(2-[3-Amino-3-fluoro-4-(isopropylamino)-1,1-bipheny...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory activity of the compound against coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50134405(CHEMBL421098 | N-(4-Carbamimidoyl-benzyl)-2-(5-iso...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory activity of the compound against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14601(CHEMBL125585 | N-[(4-carbamimidoylphenyl)methyl]-2...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory activity of the compound against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14599(CHEMBL333980 | N-[(4-carbamimidoylphenyl)methyl]-2...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory activity of the compound against coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50134405(CHEMBL421098 | N-(4-Carbamimidoyl-benzyl)-2-(5-iso...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory activity of the compound against coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM14601(CHEMBL125585 | N-[(4-carbamimidoylphenyl)methyl]-2...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory activity of the compound against coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed