Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50016729
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataKi:  8nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172802(Sodium; 8-hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oc...)
Affinity DataEC50:  114nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172817(8-Hydroxy-8-(2-pentyloxy-phenyl)-oct-5-ynoic acid ...)
Affinity DataEC50:  173nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172813(8-Hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oct-5-ynoi...)
Affinity DataEC50:  262nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172823(8-Hydroxy-8-(2-pentyloxy-phenyl)-octanoic acid met...)
Affinity DataKi:  515nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172814(8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct-5-ynoic...)
Affinity DataEC50:  549nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172805(9-Hydroxy-9-(3-pentyloxy-naphthalen-2-yl)-nonanoic...)
Affinity DataKi:  579nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172802(Sodium; 8-hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oc...)
Affinity DataEC50:  617nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172817(8-Hydroxy-8-(2-pentyloxy-phenyl)-oct-5-ynoic acid ...)
Affinity DataEC50:  642nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172816(8-Hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-oct-5-yn...)
Affinity DataKi:  695nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172806((E)-8-Hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-oct-...)
Affinity DataKi:  718nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172822(Sodium; 8-hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-...)
Affinity DataEC50:  723nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172802(Sodium; 8-hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oc...)
Affinity DataKi:  947nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172810(Sodium; 8-hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-...)
Affinity DataKi:  969nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172817(8-Hydroxy-8-(2-pentyloxy-phenyl)-oct-5-ynoic acid ...)
Affinity DataKi:  1.05E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172816(8-Hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-oct-5-yn...)
Affinity DataEC50:  1.14E+3nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172805(9-Hydroxy-9-(3-pentyloxy-naphthalen-2-yl)-nonanoic...)
Affinity DataEC50:  1.36E+3nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172813(8-Hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oct-5-ynoi...)
Affinity DataEC50:  1.41E+3nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172806((E)-8-Hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-oct-...)
Affinity DataEC50:  1.45E+3nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172810(Sodium; 8-hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-...)
Affinity DataEC50:  1.49E+3nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172805(9-Hydroxy-9-(3-pentyloxy-naphthalen-2-yl)-nonanoic...)
Affinity DataEC50:  1.53E+3nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172809(Sodium; 8-hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct...)
Affinity DataEC50:  1.54E+3nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172814(8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct-5-ynoic...)
Affinity DataEC50:  1.63E+3nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172822(Sodium; 8-hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-...)
Affinity DataKi:  4.39E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172818(Sodium; 8-hydroxy-8-(2-pentyloxy-phenyl)-octanoate...)
Affinity DataKi:  6.69E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172808(8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-octanoic ac...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172804(Sodium; 8-hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172810(Sodium; 8-hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172803((E)-8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct-5-e...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172824(9-Hydroxy-9-(2-pentyloxy-quinolin-3-yl)-nonanoic a...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172824(9-Hydroxy-9-(2-pentyloxy-quinolin-3-yl)-nonanoic a...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172823(8-Hydroxy-8-(2-pentyloxy-phenyl)-octanoic acid met...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172822(Sodium; 8-hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172804(Sodium; 8-hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172803((E)-8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct-5-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172816(8-Hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-oct-5-yn...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172823(8-Hydroxy-8-(2-pentyloxy-phenyl)-octanoic acid met...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172803((E)-8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct-5-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172824(9-Hydroxy-9-(2-pentyloxy-quinolin-3-yl)-nonanoic a...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172809(Sodium; 8-hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172820(Sodium; (E)-8-hydroxy-8-(2-pentyloxy-pyridin-3-yl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172818(Sodium; 8-hydroxy-8-(2-pentyloxy-phenyl)-octanoate...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172815(Sodium; 8-hydroxy-8-(2-pentyloxy-phenyl)-oct-5-yno...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172815(Sodium; 8-hydroxy-8-(2-pentyloxy-phenyl)-oct-5-yno...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172820(Sodium; (E)-8-hydroxy-8-(2-pentyloxy-pyridin-3-yl)...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172804(Sodium; 8-hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Cnrs Umr 6052

Curated by ChEMBL
LigandPNGBDBM50172808(8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-octanoic ac...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor alpha/Gal4 in transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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