Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50020578
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215294(2-(N-(6-chloro-7-methyl-2,3-dioxo-1,2,3,4-tetrahyd...)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215284(2-(N-(7-chloro-6-methyl-2,3-dioxo-1,2,3,4-tetrahyd...)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215283(2-(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroqui...)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215282(N-(6-chloro-7-methyl-2,3-dioxo-1,2,3,4-tetrahydroq...)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215286(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215286(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215281(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215287(N-(3-methoxybenzyl)-N-(6,7-dichloro-2,3-dioxo-1,2,...)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215296(N-(7-chloro-6-methyl-2,3-dioxo-1,2,3,4-tetrahydroq...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215285(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215276(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215281(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215281(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215279(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215298(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215297(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215292(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215280(N-(3-fluorobenzyl)-N-(6,7-dichloro-2,3-dioxo-1,2,3...)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215278(N-(6-chloro-7-ethyl-2,3-dioxo-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215277(N-(7-chloro-6-ethyl-2,3-dioxo-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 58nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215295(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215291(N-(7-chloro-6-methyl-2,3-dioxo-1,2,3,4-tetrahydroq...)
Affinity DataIC50: 74nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215288(N-(6-chloro-7-methyl-2,3-dioxo-1,2,3,4-tetrahydroq...)
Affinity DataIC50: 77nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215276(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 109nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215276(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 109nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215290(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 166nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215293(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 209nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215286(N-(6,7-dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinox...)
Affinity DataIC50: 282nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50215289(N-(7-chloro-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin...)
Affinity DataIC50: 728nMAssay Description:Antagonist activity at human NMDA NR1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed