Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50025601
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM5447(ZD1839 | N-(3-chloro-4-fluorophenyl)-7-methoxy-6-[...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247550(4-(5-Bromoindole-3-yl)-6,7-dimethoxyquinazoline | ...)
Affinity DataIC50: 131nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247551(4-(5-Chloro-6-fluoroindole-3-yl)-6,7-dimethoxyquin...)
Affinity DataIC50: 209nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247161(4-(5-Chloro-6-fluoroindole-3-yl)-7-methoxy-6-(3-mo...)
Affinity DataIC50: 333nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247160(4-(5-Chloro-6-fluoro-indole-3-yl)-6,7-di-(2-methox...)
Affinity DataIC50: 472nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247159(4-(6-Fluoro-5-methylindole-3-yl)-6,7-dimethoxyquin...)
Affinity DataIC50: 533nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM4363(alpha-Cyano-(3,4-dihydroxy)thiocinnamide | CHEMBL7...)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM4363(alpha-Cyano-(3,4-dihydroxy)thiocinnamide | CHEMBL7...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human HER2 tyrosine kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed