Compile Data Set for Download or QSAR
maximum 50k data
Found 100 Enz. Inhib. hit(s) with all data for entry = 50038582
TargetP2Y purinoceptor 6(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50118239(CHEMBL130266 | UDP | Uridine diphosphate | uridine...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271102(((((2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin...)
Affinity DataEC50:  660nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271138(CHEMBL527872 | [(2R,3S,4R,5R)-4-[(aminocarbonyl)am...)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271101(CHEMBL488132 | [(2R,3S,4R,5R)-5-(5-amino-2,4-dioxo...)
Affinity DataEC50:  610nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270555(CHEMBL505403 | {[(2R,3S,5R)-5-(2-amino-6-oxo-6,9-d...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270554(CHEMBL509434 | P1-(2-thiouridine 5'-)-P4-(2'-deoxy...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270553(CHEMBL507282 | INS-37217 | INS37217)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270552(CHEMBL476021 | P1,P4-di(uridine 5'-)beta,gamma-dic...)
Affinity DataEC50:  7.77E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270551(CHEMBL502712 | P1,P4-di(uridine 5'-)beta,gamma-dif...)
Affinity DataEC50:  2.27E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270550(CHEMBL503798 | {[(2R,3S,4R,5R)-3,4-dihydroxy-5-(2-...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50205413(CHEMBL221326 | P(1),P(4)-bis(uridin-5'-yl) tetraph...)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270549(CHEMBL503256 | P1-((2-benzyl-1,3-dioxolo-4-yl)urid...)
Affinity DataEC50:  9.97E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50241299(CHEMBL239151 | {[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,...)
Affinity DataEC50:  1.31E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270548(CHEMBL454230 | Uridine-5'-(2'-deoxy-glucose)-6'-te...)
Affinity DataEC50:  3.54E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270547(CHEMBL508122 | Uridine-5'-mannose-6'-tetraphosphat...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270546(CHEMBL444212 | Uridine-5'-galactose-1'-tetraphosph...)
Affinity DataEC50:  4.85E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270545(CHEMBL499138 | Uridine-5'-glucose-1'-tetraphosphat...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270544(CHEMBL500840 | Uridine-5'-fructose-6'-tetraphospha...)
Affinity DataEC50:  3.33E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270543(CHEMBL448985 | [({[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,...)
Affinity DataEC50:  1.88E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270542(CHEMBL474887 | Uridine-5'-cyclohexane-tetraphospha...)
Affinity DataEC50:  5.86E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270541(CHEMBL474886 | Uridine-5'-phenyl-tetraphosphate)
Affinity DataEC50:  1.89E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271292(CHEMBL482895 | Uridine-5'-alpha-glycerol-tetraphos...)
Affinity DataEC50:  1.87E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271291(CHEMBL484105 | Uridine-5'-(2-cyanoethyl)-tetraphos...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271290(CHEMBL483913 | Uridine-5'-methyl(C-P)-tetraphospha...)
Affinity DataEC50:  4.18E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271289(CHEMBL519991 | Uridine-5'-methyl-tetraphosphate)
Affinity DataEC50:  3.95E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271254(2-Thio-uridine-5'-pentaphosphate | CHEMBL482683)
Affinity DataEC50:  570nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271253(4-Thio-uridine-5'-tetraphosphate | CHEMBL521451)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271252(2-Thio-uridine-5'-tetraphosphate | CHEMBL482485)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271251(CHEMBL483502 | {[({[({[(2R,3S,4R,5R)-5-(2,4-dioxo-...)
Affinity DataEC50:  2.61E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271224(2'-C-Methyl-uridine-5'-triphosphate | CHEMBL521487)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271223(({[({[(2R,3S,4S,5R)-3,4-dihydroxy-5-(4-oxo-2-sulfa...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271222(({[({[(2R,3S,4R,5R)-4-(carbamoylamino)-5-(2,4-diox...)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271188(2-Thio-4-methylthio-uridine-5'-triphosphate | CHEM...)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271187(CHEMBL519835 | [dichloro({[({[(2R,3S,4R,5R)-3,4-di...)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271186(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(4-oxo-2-sulfa...)
Affinity DataEC50:  1.63E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50205406(((2R,3S,4R,5R)-4-amino-3-hydroxy-5-(4-oxo-2-thioxo...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50205405(({[({[(2R,3S,4R,5R)-4-amino-5-(2,4-dioxo-1,2,3,4-t...)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270555(CHEMBL505403 | {[(2R,3S,5R)-5-(2-amino-6-oxo-6,9-d...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270554(CHEMBL509434 | P1-(2-thiouridine 5'-)-P4-(2'-deoxy...)
Affinity DataEC50:  710nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270553(CHEMBL507282 | INS-37217 | INS37217)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270551(CHEMBL502712 | P1,P4-di(uridine 5'-)beta,gamma-dif...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270550(CHEMBL503798 | {[(2R,3S,4R,5R)-3,4-dihydroxy-5-(2-...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50205413(CHEMBL221326 | P(1),P(4)-bis(uridin-5'-yl) tetraph...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50241299(CHEMBL239151 | {[(2R,3S,4R,5R)-5-(2,4-dioxo-1,2,3,...)
Affinity DataEC50:  870nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270548(CHEMBL454230 | Uridine-5'-(2'-deoxy-glucose)-6'-te...)
Affinity DataEC50:  4.32E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270547(CHEMBL508122 | Uridine-5'-mannose-6'-tetraphosphat...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270546(CHEMBL444212 | Uridine-5'-galactose-1'-tetraphosph...)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270545(CHEMBL499138 | Uridine-5'-glucose-1'-tetraphosphat...)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270544(CHEMBL500840 | Uridine-5'-fructose-6'-tetraphospha...)
Affinity DataEC50:  6.30E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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