Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50027217
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]MK912 from human cloned adrenergic alpha2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  275nMAssay Description:Inhibition of cloned adrenergic alpha1D receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [125I]-APT from histamine H2 receptor in brain of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]SMT from histamine H3 receptor in forebrain of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataIC50:  185nMAssay Description:Displacement of [3H]MK912 from human cloned adrenergic alpha2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataIC50:  560nMAssay Description:Inhibition of cloned adrenergic alpha1D receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataIC50:  1.25E+3nMAssay Description:Displacement of [125I]-APT from histamine H2 receptor in brain of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataIC50:  2.35E+3nMAssay Description:Displacement of [3H]SMT from histamine H3 receptor in forebrain of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed