Affinity DataKi: 69nMAssay Description:Displacement of [3H]MK912 from human cloned adrenergic alpha2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Inhibition of cloned adrenergic alpha1D receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Displacement of [125I]-APT from histamine H2 receptor in brain of guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Displacement of [3H]SMT from histamine H3 receptor in forebrain of ratMore data for this Ligand-Target Pair
Affinity DataIC50: 185nMAssay Description:Displacement of [3H]MK912 from human cloned adrenergic alpha2a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Inhibition of cloned adrenergic alpha1D receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+3nMAssay Description:Displacement of [125I]-APT from histamine H2 receptor in brain of guinea pigMore data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+3nMAssay Description:Displacement of [3H]SMT from histamine H3 receptor in forebrain of ratMore data for this Ligand-Target Pair