Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50028524
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267395(5'-chloro-5'-deoxy-N6-((-endo-norborn-2-yl)adenosi...)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267577(N6-((+/-)-endo-norborn-2-yl)adenosine | CHEMBL4896...)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267393(N6-Cyclopentyl-9H-(5-chloro-5-deoxy-beta-D-ribofur...)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267578(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(beta-D-ribofu...)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267394(2,5'-dichloro-5'-deoxy-N6-cyclopentyladenosine | C...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267396(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(5-chloro-5-de...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267575(N6-(+/-)-endo-Norbornyl-9H-(2-C-methyl-beta-D-ribo...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267576(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(2-C-methyl-be...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267475(N6-(+/-)-endo-Norbornyl-9H-(2-C-methyl-5-chloro-5-...)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267476(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(2-C-methyl-5-...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267474(2-Chloro-N6-cyclopentyl-9H-(2-C-methyl-5-chloro-5-...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267397(N6-Cyclopentyl-9H-(2-C-methyl-5-chloro-5-deoxy-bet...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267477(N6-cyclopentyl-5'-(2-fluorophenylthio)-5'-deoxyade...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267577(N6-((+/-)-endo-norborn-2-yl)adenosine | CHEMBL4896...)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267578(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(beta-D-ribofu...)
Affinity DataKi:  129nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267574(N6-Tetrahydrofuranyl-9H-[5-deoxy-5-(2-fluorophenyl...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267478(2-Chloro-N6-cyclopentyl-9H-[5-deoxy-5-(2-fluorophe...)
Affinity DataKi:  258nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267477(N6-cyclopentyl-5'-(2-fluorophenylthio)-5'-deoxyade...)
Affinity DataKi:  296nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267393(N6-Cyclopentyl-9H-(5-chloro-5-deoxy-beta-D-ribofur...)
Affinity DataKi:  376nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267394(2,5'-dichloro-5'-deoxy-N6-cyclopentyladenosine | C...)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267478(2-Chloro-N6-cyclopentyl-9H-[5-deoxy-5-(2-fluorophe...)
Affinity DataKi:  479nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267574(N6-Tetrahydrofuranyl-9H-[5-deoxy-5-(2-fluorophenyl...)
Affinity DataKi:  746nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267578(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(beta-D-ribofu...)
Affinity DataKi:  797nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267393(N6-Cyclopentyl-9H-(5-chloro-5-deoxy-beta-D-ribofur...)
Affinity DataKi:  837nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267536(N6-(+/-)-endo-Norbornyl-9H-[2-C-methyl-5-deoxy-5-(...)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267535(2-Chloro-N6-cyclopentyl-9H-[2-C-methyl-5-deoxy-5-(...)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267577(N6-((+/-)-endo-norborn-2-yl)adenosine | CHEMBL4896...)
Affinity DataKi:  1.27E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267395(5'-chloro-5'-deoxy-N6-((-endo-norborn-2-yl)adenosi...)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267395(5'-chloro-5'-deoxy-N6-((-endo-norborn-2-yl)adenosi...)
Affinity DataKi:  1.34E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267396(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(5-chloro-5-de...)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267534(N6-Cyclopentyl-9H-[2-C-methyl-5-deoxy-5-(2-fluorop...)
Affinity DataKi:  1.44E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267534(N6-Cyclopentyl-9H-[2-C-methyl-5-deoxy-5-(2-fluorop...)
Affinity DataKi:  1.68E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267396(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(5-chloro-5-de...)
Affinity DataKi:  2.05E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267535(2-Chloro-N6-cyclopentyl-9H-[2-C-methyl-5-deoxy-5-(...)
Affinity DataKi:  2.15E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267394(2,5'-dichloro-5'-deoxy-N6-cyclopentyladenosine | C...)
Affinity DataKi:  2.16E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267478(2-Chloro-N6-cyclopentyl-9H-[5-deoxy-5-(2-fluorophe...)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267575(N6-(+/-)-endo-Norbornyl-9H-(2-C-methyl-beta-D-ribo...)
Affinity DataKi:  2.52E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267395(5'-chloro-5'-deoxy-N6-((-endo-norborn-2-yl)adenosi...)
Affinity DataKi:  2.74E+3nMAssay Description:Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267537(2-Chloro-N6-(+/-)-endo-norbornyl-9H-[2-C-methyl-5-...)
Affinity DataKi:  2.97E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267474(2-Chloro-N6-cyclopentyl-9H-(2-C-methyl-5-chloro-5-...)
Affinity DataKi:  3.03E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267393(N6-Cyclopentyl-9H-(5-chloro-5-deoxy-beta-D-ribofur...)
Affinity DataKi:  3.21E+3nMAssay Description:Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267536(N6-(+/-)-endo-Norbornyl-9H-[2-C-methyl-5-deoxy-5-(...)
Affinity DataKi:  3.48E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267537(2-Chloro-N6-(+/-)-endo-norbornyl-9H-[2-C-methyl-5-...)
Affinity DataKi:  4.35E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267576(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(2-C-methyl-be...)
Affinity DataKi:  4.49E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267394(2,5'-dichloro-5'-deoxy-N6-cyclopentyladenosine | C...)
Affinity DataKi:  4.83E+3nMAssay Description:Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267577(N6-((+/-)-endo-norborn-2-yl)adenosine | CHEMBL4896...)
Affinity DataKi:  4.93E+3nMAssay Description:Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267477(N6-cyclopentyl-5'-(2-fluorophenylthio)-5'-deoxyade...)
Affinity DataKi:  5.17E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267476(2-Chloro-N6-(+/-)-endo-norbornyl-9H-(2-C-methyl-5-...)
Affinity DataKi:  5.90E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267397(N6-Cyclopentyl-9H-(2-C-methyl-5-chloro-5-deoxy-bet...)
Affinity DataKi:  6.74E+3nMAssay Description:Displacement of [3H]HEMADO from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267575(N6-(+/-)-endo-Norbornyl-9H-(2-C-methyl-beta-D-ribo...)
Affinity DataKi:  8.78E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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