Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50004360
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482153BDBM50482153(CHEMBL1098750)
Affinity DataIC50: 32nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482154BDBM50482154(CHEMBL1095415)
Affinity DataIC50: 32nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482145BDBM50482145(CHEMBL1098070)
Affinity DataIC50: 46nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482150BDBM50482150(CHEMBL1094396)
Affinity DataIC50: 59nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482157BDBM50482157(CHEMBL1097709)
Affinity DataIC50: 72nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482151BDBM50482151(CHEMBL1098435)
Affinity DataIC50: 75nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482149BDBM50482149(CHEMBL1097708)
Affinity DataIC50: 237nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482156BDBM50482156(CHEMBL1098436)
Affinity DataIC50: 300nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482148BDBM50482148(CHEMBL1097710)
Affinity DataIC50: 374nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482152BDBM50482152(CHEMBL1095649)
Affinity DataIC50: 385nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482147BDBM50482147(CHEMBL1096709)
Affinity DataIC50: 757nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482155BDBM50482155(CHEMBL1096708)
Affinity DataIC50: 876nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482146BDBM50482146(CHEMBL1096966)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482158BDBM50482158(CHEMBL1096035)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PDE4 in human U937 cells after 30 mins by electrochemiluminescence based immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed