Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50031882
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320966(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320954(3-((4-(6-Methylpyridin-2-yl)-3-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50252542(3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320953(3-((4-(6-Methylpyridin-2-yl)-3-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  61nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320958(3-((3-(6-Methylpyridin-2-yl)-4-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320952(6-(2-tert-butyl-5-(6-methylpyridin-2-yl)-1H-imidaz...)
Affinity DataIC50:  162nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50298220(2-(4-(benzo[d][1,3]dioxol-5-yl)-2-tert-butyl-1H-im...)
Affinity DataIC50:  169nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320962(3-((3-(6-Methylpyridin-2-yl)-4-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  231nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320956(3-((3-(6-Methylpyridin-2-yl)-4-(1,5-naphthyridin-2...)
Affinity DataIC50:  255nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320960(3-((3-(6-Methylpyridin-2-yl)-4-(1,5-naphthyridin-2...)
Affinity DataIC50:  318nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  540nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  650nMAssay Description:Inhibition of PKCmuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  940nMAssay Description:Inhibition of VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320965(3-((5-(6-Methylpyridin-2-yl)-4-(1,5-naphthyridin-2...)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320963(3-((5-(6-Methylpyridin-2-yl)-4-(1,5-naphthyridin-2...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320955(3-((5-(6-Methylpyridin-2-yl)-4-(1,5-naphthyridin-2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320957(3-((5-(6-Methylpyridin-2-yl)-4-(quinolin-6-yl)-1H-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320961(3-((5-(6-Methylpyridin-2-yl)-4-(quinolin-6-yl)-1H-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320959(3-((5-(6-Methylpyridin-2-yl)-4-(1,5-naphthyridin-2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed