Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50032238
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279431(3-(4-Chloro-phenyl)-2-[2-(4-chloro-phenylamino)-4-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of PMA-induced transcriptional activation treated 24 hrs before PMA challenge by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279429(3-(4-Chloro-phenyl)-2-(4-methyl-2-methylamino-thia...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of PMA-induced transcriptional activation treated 24 hrs before PMA challenge by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50326123(3-(4-Chloro-phenyl)-2-[2-(4-chloro-phenylamino)-4-...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of PMA-induced transcriptional activation treated 24 hrs before PMA challenge by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50326119(CHEMBL1242070 | [5-(4-Oxo-3-phenyl-3,4-dihydro-qui...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of PMA-induced transcriptional activation treated 24 hrs before PMA challenge by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50326121(CHEMBL1242520 | {5-[3-(4-Chloro-phenyl)-4-oxo-3,4-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of PMA-induced transcriptional activation treated 24 hrs before PMA challenge by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50326120(2-[2-(4-Chloro-phenylamino)-4-phenyl-thiazol-5-yl]...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of PMA-induced transcriptional activation treated 24 hrs before PMA challenge by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50326122(3-(4-Chloro-phenyl)-2-(2-methylamino-4-phenyl-thia...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of PMA-induced transcriptional activation treated 24 hrs before PMA challenge by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed