Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50004651
TargetATP-dependent translocase ABCB1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50485270(CHEMBL2042913)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of p-glycoprotein expressed in human MCF-7/DX1 cells assessed as accumulation of calcein-AM by FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50485269(CHEMBL2042912)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of p-glycoprotein expressed in human MCF-7/DX1 cells assessed as accumulation of calcein-AM by FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50485274(CHEMBL2042911)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of p-glycoprotein expressed in human MCF-7/DX1 cells assessed as accumulation of calcein-AM by FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50485272(CHEMBL2042909)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of p-glycoprotein expressed in human MCF-7/DX1 cells assessed as accumulation of calcein-AM by FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50485271(CHEMBL2042914)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of p-glycoprotein expressed in human MCF-7/DX1 cells assessed as accumulation of calcein-AM by FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50485273(CHEMBL2042910)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of p-glycoprotein expressed in human MCF-7/DX1 cells assessed as accumulation of calcein-AM by FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50485267(CHEMBL2042907)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of p-glycoprotein expressed in human MCF-7/DX1 cells assessed as accumulation of calcein-AM by FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50485268(CHEMBL2042908)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of p-glycoprotein expressed in human MCF-7/DX1 cells assessed as accumulation of calcein-AM by FACS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed