Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50042964
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433865BDBM50433865(CHEMBL2380402)
Affinity DataKi:  4nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433878BDBM50433878(CHEMBL2380389)
Affinity DataKi:  6nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433880BDBM50433880(CHEMBL2380387)
Affinity DataKi:  6.20nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433864BDBM50433864(CHEMBL2380403)
Affinity DataKi:  6.60nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433877BDBM50433877(CHEMBL2380390)
Affinity DataKi:  7nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433871BDBM50433871(CHEMBL2380396)
Affinity DataKi:  10nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433877BDBM50433877(CHEMBL2380390)
Affinity DataKi:  11nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433868BDBM50433868(CHEMBL2380400)
Affinity DataKi:  11nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433878BDBM50433878(CHEMBL2380389)
Affinity DataKi:  12nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433866BDBM50433866(CHEMBL2380314)
Affinity DataKi:  21nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433872BDBM50433872(CHEMBL2380395)
Affinity DataKi:  31nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433872BDBM50433872(CHEMBL2380395)
Affinity DataKi:  31nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433879BDBM50433879(CHEMBL2380388)
Affinity DataKi:  50nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433867BDBM50433867(CHEMBL2380401)
Affinity DataKi:  62nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433875BDBM50433875(CHEMBL2380392)
Affinity DataKi:  68nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433879BDBM50433879(CHEMBL2380388)
Affinity DataKi:  70nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433880BDBM50433880(CHEMBL2380387)
Affinity DataKi:  91nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433881BDBM50433881(CHEMBL2380406)
Affinity DataKi:  230nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433881BDBM50433881(CHEMBL2380406)
Affinity DataKi:  310nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433873BDBM50433873(CHEMBL2380394)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433865BDBM50433865(CHEMBL2380402)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433874BDBM50433874(CHEMBL2380393)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433864BDBM50433864(CHEMBL2380403)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433882BDBM50433882(CHEMBL2380405)
Affinity DataKi:  4.10E+3nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433869BDBM50433869(CHEMBL2380398)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433866BDBM50433866(CHEMBL2380314)
Affinity DataKi: >1.20E+4nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433869BDBM50433869(CHEMBL2380398)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433867BDBM50433867(CHEMBL2380401)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433876BDBM50433876(CHEMBL2380391)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433876BDBM50433876(CHEMBL2380391)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433868BDBM50433868(CHEMBL2380400)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433871BDBM50433871(CHEMBL2380396)
Affinity DataKi:  3.60E+4nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433874BDBM50433874(CHEMBL2380393)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433863BDBM50433863(CHEMBL2380404)
Affinity DataKi:  8.50E+4nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433872BDBM50433872(CHEMBL2380395)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433872BDBM50433872(CHEMBL2380395)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433863BDBM50433863(CHEMBL2380404)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433875BDBM50433875(CHEMBL2380392)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433870BDBM50433870(CHEMBL2380397)
Affinity DataKi: >2.00E+5nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433876BDBM50433876(CHEMBL2380391)
Affinity DataKi: >2.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433883BDBM50433883(CHEMBL2380399)
Affinity DataKi: >2.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433876BDBM50433876(CHEMBL2380391)
Affinity DataKi: >2.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433870BDBM50433870(CHEMBL2380397)
Affinity DataKi: >2.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrilysin(Human)
Florida State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433883BDBM50433883(CHEMBL2380399)
Affinity DataKi: >2.00E+5nMAssay Description:Inhibition of MMP-7 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed