Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 7148
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM18050(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)
Affinity DataIC50:  18nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM178023(4-[2-(2,4-Diamino-5,6,7,8-tetrahydropyrido[3,2-d]p...)
Affinity DataIC50:  40nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM178024(4-[2-(2,4-Diamino-5-formyl-5,6,7,8-tetrahydropyrid...)
Affinity DataIC50:  41nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM178027(4-[2-(2-Diamino-4-hydroxy-5,6,7,8-tetrahydropyrido...)
Affinity DataIC50:  59nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM178029(4-[2-(2-Amino-4-hydroxy-5-allyl-5,6,7,8-tetrahydro...)
Affinity DataIC50:  298nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM178030(N-[4-[2-(2,4-Diamino-5-formyl-5,6,7,8-tetrahydropy...)
Affinity DataIC50:  590nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM178026(4-[2-[2,4-Diamino-5-(2,3-dibromopropyl)-5,6,7,8-te...)
Affinity DataIC50:  680nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM178025(4-[2-(2,4-Diamino-5-allyl-5,6,7,8-tetrahydropyrido...)
Affinity DataIC50:  706nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Peking University

LigandPNGBDBM178028(4-[2-(2-Amino-4-hydroxy-5-formyl-5,6,7,8- tetrahyd...)
Affinity DataIC50:  1.01E+4nMpH: 7.5Assay Description:The recombinant human (rh) DHFR was purchased from Sigma-Aldrich (Shanghai, China). All rhDHFR enzymes were assayed spectrophotometrically in a solut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed