Found 22 Enz. Inhib. hit(s) with all data for entry = 50006548 
Affinity DataEC50: 71nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 209nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Activity at CB1R in mouse brain membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding preincubated for 60 mins prior to [35S]GT...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Positive allosteric modulator activity at human CB1R expressed in CHO cells assessed as enhanced binding of [3H]CP55,940 after 60 mins by liquid scin...More data for this Ligand-Target Pair
Affinity DataEC50: 324nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataEC50: 4.90nMAssay Description:Positive allosteric modulator activity at human CB1R expressed in CHO cells assessed as enhanced binding of [3H]CP55,940 after 60 mins by liquid scin...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 166nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 1.12E+3nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 389nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 683nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 64nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Affinity DataEC50: 118nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 83nMAssay Description:Positive allosteric modulator activity at human CB1R expressed in CHO cells assessed as enhanced binding of [3H]CP55,940 after 60 mins by liquid scin...More data for this Ligand-Target Pair
Affinity DataEC50: 174nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
