Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50047168
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Max Planck Institute For Molecular Genetics

Curated by ChEMBL
LigandPNGBDBM50151924(CHEMBL3781424)
Affinity DataKi:  700nMAssay Description:Competitive binding affinity to PPARgamma (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Max Planck Institute For Molecular Genetics

Curated by ChEMBL
LigandPNGBDBM50151924(CHEMBL3781424)
Affinity DataKi:  5.20E+3nMAssay Description:Competitive binding affinity to PPARbeta/delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Max Planck Institute For Molecular Genetics

Curated by ChEMBL
LigandPNGBDBM50151924(CHEMBL3781424)
Affinity DataKi:  9.10E+3nMAssay Description:Competitive binding affinity to PPARalpha (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed