Found 40 Enz. Inhib. hit(s) with all data for entry = 50001467 
Affinity DataKi: 0.150nMAssay Description:Binding affinity to Mu-type opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity to delta-type opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.252nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Displacement of [125I]-DAMGO from mouse FLAG-tagged Mu-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma counting analys...More data for this Ligand-Target Pair
Affinity DataIC50: 0.350nMAssay Description:Compound was tested for inhibition of hog kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:Displacement of [125I]-DAMGO from mouse FLAG-tagged Mu-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma counting analys...More data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:The compound was tested for inhibition of rat plasma renin at pH of 6.0.More data for this Ligand-Target Pair
Affinity DataIC50: 0.760nMAssay Description:Displacement of [125I]-DAMGO from mouse FLAG-tagged Mu-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma counting analys...More data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:The compound was tested for inhibition of rabbit plasma renin.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]-Deltorphin II from mouse FLAG-tagged delta-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma coun...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]-DAMGO from mouse FLAG-tagged Mu-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma counting analys...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Displacement of [125I]-DAMGO from mouse FLAG-tagged Mu-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma counting analys...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Displacement of [125I]-Deltorphin II from mouse FLAG-tagged delta-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma coun...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125I]-DAMGO from mouse FLAG-tagged Mu-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma counting analys...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity to Mu-type opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Compound was tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Displacement of [3H][Ile5,6]-deltorphin II from delta-type opioid receptor in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of Angiotensin I converting enzyme in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Agonist activity at mu-opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically induced contractions after 3 mins post doseMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]-CTOP from Mu-type opioid receptor in Sprague-Dawley rat brain homogenate after 180 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Displacement of [125I]-Deltorphin II from mouse FLAG-tagged delta-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma coun...More data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 153nMAssay Description:Displacement of [125I]-Deltorphin II from mouse FLAG-tagged delta-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma coun...More data for this Ligand-Target Pair
Affinity DataIC50: 167nMAssay Description:Displacement of [125I]-Deltorphin II from mouse FLAG-tagged delta-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma coun...More data for this Ligand-Target Pair
Affinity DataIC50: 263nMAssay Description:Agonist activity at delta-type opioid receptor in ICR mouse vas deferens assessed as potentiation of electrically stimulated contractions after 3 min...More data for this Ligand-Target Pair
Affinity DataIC50: 295nMAssay Description:Binding affinity to delta-type opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Displacement of [125I]-Deltorphin II from mouse FLAG-tagged delta-type opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma coun...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:Displacement of [H][p-ClPhe4]-DPDPE from delta-type opioid receptor in Sprague-Dawley rat brain homogenates after 180 mins by scintillation countingMore data for this Ligand-Target Pair
