Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50022490
Affinity DataKi: 65nMAssay Description:Competitive inhibition of PRDM9 (unknown origin) assessed as inhibition constant in presence of varying concentration of SAM and peptide substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of PRDM9 (unknown origin) (195 to 415 residues) using biotin-tagged Histone H3 (1 to 25) and 3H-SAM as substrate incubated for 30 mins by ...More data for this Ligand-Target Pair
Affinity DataKd: 87nMAssay Description:Binding affinity to PRDM9 (unknown origin) (195 to 415 residues) assessed as dissociation constant measured at 60 to 120 secs in presence of SAM by b...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of FLAG tagged PRDM9 transfected in HEK293T cells assessed as reduction in trimethylation of ectopic H3K4 measured after 20 hrs by Western...More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of PRDM7 (unknown origin) using biotin-tagged Histone H3 (1 to 25) and 3H-SAM as substrate incubated for 90 mins by topcount plate reader ...More data for this Ligand-Target Pair
