Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50020526
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50630845(CHEMBL5435819)
Affinity DataIC50: 1nMAssay Description:Inhibition of human BCR-ABL1 M351T mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human BCR-ABL1 Q252H mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50630845(CHEMBL5435819)
Affinity DataIC50: 1nMAssay Description:Inhibition of human BCR-ABL1 H396P mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human BCR-ABL1 M351T mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human BCR-ABL1 Y253F mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50630845(CHEMBL5435819)
Affinity DataIC50: 1nMAssay Description:Inhibition of human BCR-ABL1 Q252H mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50630845(CHEMBL5435819)
Affinity DataIC50: 1nMAssay Description:Inhibition of human BCR-ABL1 Y253F mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50630845(CHEMBL5435819)
Affinity DataIC50: 1nMAssay Description:Inhibition of human wild type BCR-ABL1 by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human BCR-ABL1 H396P mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human wild type BCR-ABL1 by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50630845(CHEMBL5435819)
Affinity DataIC50: 2nMAssay Description:Inhibition of human wild type c-Src by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human wild type c-Src by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 44nMAssay Description:Inhibition of human BCR-ABL1 T315I mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Georgia

Curated by ChEMBL
LigandPNGBDBM50630845(CHEMBL5435819)
Affinity DataIC50: 47nMAssay Description:Inhibition of human BCR-ABL1 T315I mutant by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed