Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50009476
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50053929(CHEMBL88147 | N-(9-Chloro-2-furan-2-yl-[1,2,4]tria...)
Affinity DataKi:  0.650nMAssay Description:In vitro binding affinity against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50059376(9-Methyl-2-phenyl-5,9-dihydro-[1,2,4]triazolo[5,1-...)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50059375(5-Amino-3-(4-methoxy-phenyl)-thiazolo[3,2-a]pyrimi...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50053924(3,6-Dichloro-2-(2-isopropoxy-4-methyl-phenyl)-chro...)
Affinity DataKi:  560nMAssay Description:In vitro binding affinity against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50084018(2-Phenylacetylamino-4,7-dihydro-5H-thieno[2,3-c]py...)
Affinity DataKi:  600nMAssay Description:In vitro binding affinity against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50084019(6,7-Dimethoxy-3-[4-(4-methoxy-phenyl)-thiazol-2-yl...)
Affinity DataKi:  1.30E+3nMAssay Description:In vitro binding affinity against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50084017(CHEMBL326389 | {[(2-Benzoylamino-5-bromo-phenyl)-p...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding stimulated by 20 uM 5''-N-ethyluronamidoadenosine (NECA) in membranes of HEK-293 cells expressing human Adeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50084018(2-Phenylacetylamino-4,7-dihydro-5H-thieno[2,3-c]py...)
Affinity DataIC50:  186nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding stimulated by 20 uM 5''-N-ethyluronamidoadenosine (NECA) in membranes of HEK-293 cells expressing human Adeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50084019(6,7-Dimethoxy-3-[4-(4-methoxy-phenyl)-thiazol-2-yl...)
Affinity DataIC50:  255nMAssay Description:In vitro binding affinity against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Chembridge

Curated by ChEMBL
LigandPNGBDBM50084017(CHEMBL326389 | {[(2-Benzoylamino-5-bromo-phenyl)-p...)
Affinity DataIC50:  407nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding stimulated by 5 uM 5''-N-ethyluronamidoadenosine (NECA) in membranes of HEK-293 cells expressing human Adenos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed