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Found 32 Enz. Inhib. hit(s) with all data for entry = 50014206
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573588(CHEMBL4871554)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573589(CHEMBL4864883)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573587(CHEMBL4861092)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452336(CHEMBL2113406)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50205709((2R,3R,4S,5R)-2-(6-amino-2-(phenylethynyl)-9H-puri...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452335(CHEMBL2113484)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452335(CHEMBL2113484)
Affinity DataKi:  79nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50205709((2R,3R,4S,5R)-2-(6-amino-2-(phenylethynyl)-9H-puri...)
Affinity DataKi:  646nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573587(CHEMBL4861092)
Affinity DataKi:  803nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50366687(CHEMBL3350497 | CHEMBL611516)
Affinity DataKi:  856nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452336(CHEMBL2113406)
Affinity DataKi:  864nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573591(CHEMBL4847237)
Affinity DataKi:  879nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50205709((2R,3R,4S,5R)-2-(6-amino-2-(phenylethynyl)-9H-puri...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cell membrane incubated for 30 mins by microplate beta scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573593(CHEMBL4855141)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573588(CHEMBL4871554)
Affinity DataKi:  1.38E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK cell membrane incubated for 30 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573592(CHEMBL4852007)
Affinity DataKi:  1.94E+3nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573591(CHEMBL4847237)
Affinity DataKi:  1.99E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cell membrane incubated for 30 mins by microplate beta scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452335(CHEMBL2113484)
Affinity DataKi:  2.05E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cell membrane incubated for 30 mins by microplate beta scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573587(CHEMBL4861092)
Affinity DataKi:  3.33E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK cell membrane incubated for 30 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573589(CHEMBL4864883)
Affinity DataKi:  3.34E+3nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573587(CHEMBL4861092)
Affinity DataKi:  7.10E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cell membrane incubated for 30 mins by microplate beta scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573592(CHEMBL4852007)
Affinity DataKi:  8.61E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573590(CHEMBL4873585)
Affinity DataKi:  8.77E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in HeLa cell membrane incubated for 180 mins by microplate beta scintillation cou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573590(CHEMBL4873585)
Affinity DataKi:  1.33E+4nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573588(CHEMBL4871554)
Affinity DataIC50:  1.46E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452335(CHEMBL2113484)
Affinity DataIC50:  2.03E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573589(CHEMBL4864883)
Affinity DataIC50:  2.20E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573587(CHEMBL4861092)
Affinity DataIC50:  2.65E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452336(CHEMBL2113406)
Affinity DataIC50:  7.41E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells by beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573587(CHEMBL4861092)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human adenosine A3 receptor transfected in CHO cells assessed as cAMP level measured after 35 mins by cAMP enzyme immunoassayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50452336(CHEMBL2113406)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human adenosine A3 receptor transfected in CHO cells assessed as cAMP level measured after 35 mins by cAMP enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Institute Of Medical Biology Pas

Curated by ChEMBL
LigandPNGBDBM50573589(CHEMBL4864883)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human adenosine A3 receptor transfected in CHO cells assessed as cAMP level measured after 35 mins by cAMP enzyme immunoassayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed