Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50035138
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101904(CHEMBL52741 | GDP-Azasugar analogue)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of GnRH-stimulated luteinizing hormone (LH) release in rat pituitary cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM92459(CHEMBL384759 | GDP | Guanosine Diphosphate)
Affinity DataIC50:  6.70E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101904(CHEMBL52741 | GDP-Azasugar analogue)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101907(({[(2R,3S,4R,5R)-5-(2-azaniumyl-6-hydroxy-9H-purin...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101906(CHEMBL53188 | GDP-Azasugar analogue)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed