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Found 12 Enz. Inhib. hit(s) with all data for entry = 50035245
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116818(4-Sulfamoyloxy-benzoic acid heptyl ester | CHEMBL4...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116815(4-Sulfamoyloxy-benzoic acid hexyl ester | CHEMBL78...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116813(4-Sulfamoyloxy-benzoic acid nonyl ester | CHEMBL80...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116814(4-Sulfamoyloxy-benzoic acid octyl ester | CHEMBL42...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116811(4-Sulfamoyloxy-benzoic acid pentyl ester | CHEMBL3...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116810(4-Sulfamoyloxy-benzoic acid butyl ester | CHEMBL76...)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50051829(4-methyl-2-oxo-2H-chromen-7-yl sulfamate | CHEMBL1...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116817(4-Sulfamoyloxy-benzoic acid propyl ester | CHEMBL7...)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116812(4-Sulfamoyloxy-benzoic acid decyl ester | CHEMBL30...)
Affinity DataIC50:  2.24E+4nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116819(4-Sulfamoyloxy-benzoic acid methyl ester | CHEMBL3...)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibitory activity against Estrone sulfatase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Kingston University

Curated by ChEMBL
LigandPNGBDBM50116816(4-Sulfamoyloxy-benzoic acid ethyl ester | CHEMBL79...)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibitory activity against Estrone SulfataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed