Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with all data for entry = 50035728
TargetDihydrofolate reductase(Mus musculus (Mouse))
Institute

Curated by ChEMBL
LigandPNGBDBM50367055(4-Aminofolic acid | 4-Aminopteroic acid | AMINOPTE...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR) isolated from L1210 murine leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Mus musculus (Mouse))
Institute

Curated by ChEMBL
LigandPNGBDBM50023405(3-(Carboxymethyl-{4-[(2,4-diamino-pteridin-6-ylmet...)
Affinity DataIC50:  38nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Mus musculus (Mouse))
Institute

Curated by ChEMBL
LigandPNGBDBM50023404(5-{4-[(2,4-Diamino-pteridin-6-ylmethyl)-methyl-ami...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Mus musculus (Mouse))
Institute

Curated by ChEMBL
LigandPNGBDBM50023406(5-{4-[(2,4-Diamino-pteridin-6-ylmethyl)-amino]-ben...)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Mus musculus (Mouse))
Institute

Curated by ChEMBL
LigandPNGBDBM50023408(2-{3-[(2,4-Diamino-pteridin-6-ylmethyl)-amino]-ben...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR) isolated from L1210 murine leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed