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Found 43 Enz. Inhib. hit(s) with all data for entry = 50039387
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336890((+/-)-N-(2-(benzhydrylsulfinyl)ethyl)-3-phenylprop...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336890((+/-)-N-(2-(benzhydrylsulfinyl)ethyl)-3-phenylprop...)
Affinity DataKi:  194nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  286nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336891((+/-)-2-(Bis(4-chlorophenyl)methylsulfinyl)-N,N-di...)
Affinity DataKi:  406nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336899((+/-)-2-(Bis(4-bromophenyl)methylsulfinyl)acetamid...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336898((+/-)-2-(Bis(4-chlorophenyl)methylsulfinyl)acetami...)
Affinity DataKi:  919nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336894(2-(Bis(4-fluorophenyl)methylthio)acetamide | CHEMB...)
Affinity DataKi:  1.57E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336907((+/-)-2-(Bis(4-bromophenyl)methylsulfinyl)-N-methy...)
Affinity DataKi:  1.65E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336896(2-(Bis(4-bromophenyl)methylthio)acetamide | CHEMBL...)
Affinity DataKi:  1.93E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336897((+/-)-2-(Bis(4-fluorophenyl)methylsulfinyl)acetami...)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336896(2-(Bis(4-bromophenyl)methylthio)acetamide | CHEMBL...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336895(2-(Bis(4-chlorophenyl)methylthio)acetamide | CHEMB...)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336890((+/-)-N-(2-(benzhydrylsulfinyl)ethyl)-3-phenylprop...)
Affinity DataKi:  2.35E+3nMAssay Description:Displacement of [3H]nisoxetine from NET in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336906((+/-)-2-(Bis(4-chlorophenyl)methylsulfinyl)-N-meth...)
Affinity DataKi:  2.44E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336903(2-(Bis(4-bromophenyl)methylthio)-N,N-dimethylaceta...)
Affinity DataKi:  2.45E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50156055(2-(Diphenyl-methanesulfinyl)-acetamide | 2-(benzhy...)
Affinity DataKi:  2.52E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336908((+/-)-2-(Benzhydrylsulfinyl)-N-(3-phenylpropyl)ace...)
Affinity DataKi:  2.66E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336891((+/-)-2-(Bis(4-chlorophenyl)methylsulfinyl)-N,N-di...)
Affinity DataKi:  2.89E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336903(2-(Bis(4-bromophenyl)methylthio)-N,N-dimethylaceta...)
Affinity DataKi:  3.21E+3nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336892((R)-Modafinil | ARMODAFINIL | CHEMBL1201192 | Nuvi...)
Affinity DataKi:  3.26E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [3H]nisoxetine from NET in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336902(2-(Bis(4-chlorophenyl)methylthio)-N,N-dimethylacet...)
Affinity DataKi:  4.51E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336902(2-(Bis(4-chlorophenyl)methylthio)-N,N-dimethylacet...)
Affinity DataKi:  5.98E+3nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336893((S)-Modafinil | CHEMBL1672355)
Affinity DataKi:  7.64E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336901(2-(Bis(4-fluorophenyl)methylthio)-N,N-dimethylacet...)
Affinity DataKi:  9.51E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336899((+/-)-2-(Bis(4-bromophenyl)methylsulfinyl)acetamid...)
Affinity DataKi:  1.06E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336895(2-(Bis(4-chlorophenyl)methylthio)acetamide | CHEMB...)
Affinity DataKi:  1.27E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336905((+/-)-2-(Bis(4-bromophenyl)methylsulfinyl)-N,N-dim...)
Affinity DataKi:  1.42E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336909((+/-)-2-(Bis(4-fluorophenyl)methylsulfinyl)-N,N-di...)
Affinity DataKi:  1.62E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336900(2-(Benzhydrylthio)-N,N-dimethylacetamide | CHEMBL1...)
Affinity DataKi:  1.65E+4nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336903(2-(Bis(4-bromophenyl)methylthio)-N,N-dimethylaceta...)
Affinity DataKi:  1.92E+4nMAssay Description:Displacement of [3H]nisoxetine from NET in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336905((+/-)-2-(Bis(4-bromophenyl)methylsulfinyl)-N,N-dim...)
Affinity DataKi:  2.13E+4nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336904((+/-)-2-(Bis(4-chlorophenyl)methylsulfinyl)-N,N-di...)
Affinity DataKi:  2.23E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336901(2-(Bis(4-fluorophenyl)methylthio)-N,N-dimethylacet...)
Affinity DataKi:  2.59E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336907((+/-)-2-(Bis(4-bromophenyl)methylsulfinyl)-N-methy...)
Affinity DataKi:  3.32E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336904((+/-)-2-(Bis(4-chlorophenyl)methylsulfinyl)-N,N-di...)
Affinity DataKi:  3.46E+4nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336891((+/-)-2-(Bis(4-chlorophenyl)methylsulfinyl)-N,N-di...)
Affinity DataKi:  3.62E+4nMAssay Description:Displacement of [3H]nisoxetine from NET in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336898((+/-)-2-(Bis(4-chlorophenyl)methylsulfinyl)acetami...)
Affinity DataKi:  3.90E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336902(2-(Bis(4-chlorophenyl)methylthio)-N,N-dimethylacet...)
Affinity DataKi:  4.25E+4nMAssay Description:Displacement of [3H]nisoxetine from NET in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336910((+/-)-2-(Benzhydrylsulfinyl)-N,N-dimethylethanamin...)
Affinity DataKi:  4.58E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336895(2-(Bis(4-chlorophenyl)methylthio)acetamide | CHEMB...)
Affinity DataKi:  5.21E+4nMAssay Description:Displacement of [3H]nisoxetine from NET in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50336896(2-(Bis(4-bromophenyl)methylthio)acetamide | CHEMBL...)
Affinity DataKi:  7.77E+4nMAssay Description:Displacement of [3H]nisoxetine from NET in Sprague-Dawley rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed