Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 50046997
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142788(CHEMBL3759491)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142790(CHEMBL3759441)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142783(CHEMBL218203)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142758(CHEMBL3758881)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142754(CHEMBL26962)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50122042(CHEMBL154508 | N-(4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142787(CHEMBL3758711)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142776(CHEMBL3759607)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142786(CHEMBL3758741)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142789(CHEMBL3759865)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142794(CHEMBL3758991)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142792(CHEMBL3758610)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142753(CHEMBL3760063)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142755(CHEMBL3758913)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142791(CHEMBL3760110)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142793(CHEMBL3758665)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142784(CHEMBL3759513)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142794(CHEMBL3758991)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142785(CHEMBL3758920)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142757(CHEMBL3758368)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142795(CHEMBL3759312)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142794(CHEMBL3758991)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142760(CHEMBL3758330)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142789(CHEMBL3759865)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142758(CHEMBL3758881)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142783(CHEMBL218203)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142757(CHEMBL3758368)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142776(CHEMBL3759607)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142760(CHEMBL3758330)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142784(CHEMBL3759513)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142790(CHEMBL3759441)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142792(CHEMBL3758610)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142755(CHEMBL3758913)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142753(CHEMBL3760063)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142757(CHEMBL3758368)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142789(CHEMBL3759865)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50122042(CHEMBL154508 | N-(4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  104nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142795(CHEMBL3759312)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142756(CHEMBL3758403)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142791(CHEMBL3760110)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142791(CHEMBL3760110)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142792(CHEMBL3758610)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142785(CHEMBL3758920)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142754(CHEMBL26962)
Affinity DataKi:  168nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  186nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142790(CHEMBL3759441)
Affinity DataKi:  211nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142786(CHEMBL3758741)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50142783(CHEMBL218203)
Affinity DataKi:  238nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2S receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 68 total ) | Next | Last >>
Jump to: