Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 5865
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Merck Patent

US Patent
LigandPNGBDBM97725(US8476267, 2)
Affinity DataIC50: 22nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Merck Patent

US Patent
LigandPNGBDBM50390707(CHEMBL2070316 | US8486964, 1)
Affinity DataIC50: 26nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Merck Patent

US Patent
LigandPNGBDBM50390706(CHEMBL2070315 | US8486964, 4)
Affinity DataIC50: 46nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Rat)
Merck Patent

US Patent
LigandPNGBDBM50390706(CHEMBL2070315 | US8486964, 4)
Affinity DataIC50: 490nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
Merck Patent

US Patent
LigandPNGBDBM50390707(CHEMBL2070316 | US8486964, 1)
Affinity DataIC50: 670nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
Merck Patent

US Patent
LigandPNGBDBM50390706(CHEMBL2070315 | US8486964, 4)
Affinity DataIC50: 780nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Rat)
Merck Patent

US Patent
LigandPNGBDBM50390707(CHEMBL2070316 | US8486964, 1)
Affinity DataIC50: 930nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Rat)
Merck Patent

US Patent
LigandPNGBDBM97725(US8476267, 2)
Affinity DataIC50: 1.29E+3nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent

Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
Merck Patent

US Patent
LigandPNGBDBM97725(US8476267, 2)
Affinity DataIC50: 1.54E+3nMpH: 7.4 T: 2°CAssay Description:The 11-β-HSD-1 enzyme assay was carried out in 96 well microtiter plates in a total volume of 100 μl containing 30 mM Hepes buffer, pH 7.4 wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2013
Entry Details
US Patent