Reaction Details Report a problem with these data
Cell Reactant:
Haspin (465-798)
Syringe Reactant:
BDBM103302
Meas. Tech.:
Enzyme Inhibition
Entry Date.:
10/22/14
ΔG°:
-8.67±n/a (kcal/mole)
pH:
7.5±0
Temperature:
288.15±0 (K)
ΔH° :
-17.63±0.1 (kJ/mole)
ΔS° :
-0.03±0 (kJ/mole-K)
Citation
Chaikuad, A; Tacconi, EM; Zimmer, J; Liang, Y; Gray, NS; Tarsounas, M; Knapp, S A unique inhibitor binding site in ER K1/2 is associated with slow binding kinetics Nat Chem Biol 10:853-860 (2014) [PubMed] Article
More Info.:
Cell React
Name:
Serine/threonine-protein kinase haspin [465-798]
Synonyms:
GSG2 | HASPIN | HASP_HUMAN | Haspin (aa 465-798)
Type:
Protein
Mol. Mass.:
37973.67
Organism:
Homo sapiens (Human)
Description:
Haspin kinase domain 465-798aa (curated by PDB 4QTC)
Residue:
334
Sequence:
GECSQKGPVPFSHCLPTEKLQRCEKIGEGVFGEVFQTIADHTPVAIKIIAIEGPDLVNGSHQKTFEEILPEIIISKELSLLSGEVCNRTEGFIGLNSVHCVQGSYPPLLLKAWDHYNSTKGSANDRPDFFKDDQLFIVLEFEFGGIDLEQMRTKLSSLATAKSILHQLTASLAVAEASLRFEHRDLHWGNVLLKKTSLKKLHYTLNGKSSTIPSCGLQVSIIDYTLSRLERDGIVVFCDVSMDEDLFTGDGDYQFDIYRLMKKENNNRWGEYHPYSNVLWLHYLTDKMLKQMTFKTKCNTPAMKQIKRKIQEFHRTMLNFSSATDLLCQHSLFK