Reaction Details Report a problem with these data
Target
Kelch-like ECH-associated protein 1 [321-624]
Ligand
BDBM486703
Substrate
n/a
Meas. Tech.
Fluorescence Based Assay
Kd
<1.000±n/a nM
Citation
Barbay, JK; Chai, W; Hirst, GC; Kreutter, KD; Kummer, DA; McClure, KJ; Nishimura, RT; Shih, AY; Venable, JD; Venkatesan, H; Wei, J Inhibitors of KEAP1-Nrf2 protein-protein interaction US Patent US11427601 Publication Date 8/30/2022
More Info.:
Target
Name:
Kelch-like ECH-associated protein 1 [321-624]
Synonyms:
KEAP1 | KEAP1_PONAB | Kelch-like ECH-associated protein 1 (KEAP1)(321-624)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
33399.63
Organism:
Homo sapiens (Human)
Description:
aa 321-624
Residue:
304
Sequence:
APKVGRLIYTAGGYFRQSLSYLEAYNPSDGTWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCAPMSVPRNRIGVGVIDGHIYAVGGSHGCIHHNSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITAMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMKHRRSALGITVHQGRIYVLGGYDGHTFLDSVECYDPDTDTWSEVTRMTSGRSGVGVAVTMEPCRKQIDQQNCTC