Reaction Details Report a problem with these data
Target
Coagulation factor XIII A chain
Ligand
BDBM577483
Substrate
n/a
Meas. Tech.
Isopeptidase Assay for Estimating Inhibitor Potency
IC50
365±n/a nM
Citation
Hils, M; Pasternack, R; Büchold, C Inhibitors of blood coagulation factor XIII US Patent US11472838 Publication Date 10/18/2022
More Info.:
Target
Name:
Coagulation factor XIII A chain
Synonyms:
n/a
Type:
Protein
Mol. Mass.:
83341.88
Organism:
Pig
Description:
K7GQL2
Residue:
735
Sequence:
MAETPGTGAAFGGRRALPPNTSNAEENDPPTVELQGGLMPRGFNPQDYLNVTDVHLFKERWDSNKVDHHTDKYDSKKLIVRRGQPFYIQIDFSRPYDPRRDLFRVEYVIGRYPQENKGTYIPVPIVSELQRGKWGAKVITTEDRSVRLSVQPSPDCIVGKFRMYVAVWTPYGVIRTSRNPETDTYILFNPWCEEDAVYLDNDKEREEYVLNDIGVIFYGEFNDIKSRSWSYGQFEEGILDACLYMMDRAKMDLSGRGNPIKVSRVGSAMVNAKDDEGVLVGSWDNVYSYGVPPSAWTGSVDILLEYKSSQTPVRYGQCWVFAGVFNTFLRCLGIPARVVTNYFSAHDNNANLQLDIFLEEDGNVNSKLTKDSVWNYHCWNEAWMTRPDLPVGFGGWQVVDSTPQENSDGMYRCGPASVQAIKHGHVCFQFDAPFVFAEVNSDVIYITAKKDGTHVVKTLDTTHIGKLIVTKQVGADGMKDITDTYKFQEGQEEERLALETALMYGAKKPLSTEGIPKSRSDIHMDFEVERAVLGRDFKVVLTFRNNSPTRYSVTAYLSGNITFYTGVSKGEFKNETFNVTLEPLSFKTEAVWVRAGEYMGQLLEQAFLHFFVTARVNETNDVLAKQKSVVLTIPKISVKVRGTQAVGSDMVVTVEFTNPLNEPLQNVWMRLDGPGVTRPLRKIFREIRPNATVQWEEVCRPWVSGPRKLMASMTSDSLRHVYGELNLHIQRRPSV