Target
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta
Ligand
BDBM691393
Substrate
n/a
Meas. Tech.
Inhibition Activity
Kd
>10000±n/a nM
Citation
 Gray, NSTeng, MWang, EJiang, JZhang, TCantley, LCFischer, ESDonovan, KA INHIBITORS AND DEGRADERS OF PIP4K PROTEIN US Patent  US20240277852 Publication Date 8/22/2024 
Target
Name:
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta
Synonyms:
PI42B_HUMAN | PIP4K2B | PIP5K2B | Phosphatidylinositol-5-phosphate 4-kinase type-2 beta
Type:
PROTEIN
Mol. Mass.:
47382.97
Organism:
Human
Description:
ChEMBL_774395
Residue:
416
Sequence:
MSSNCTSTTAVAVAPLSASKTKTKKKHFVCQKVKLFRASEPILSVLMWGVNHTINELSNVPVPVMLMPDDFKAYSKIKVDNHLFNKENLPSRFKFKEYCPMVFRNLRERFGIDDQDYQNSVTRSAPINSDSQGRCGTRFLTTYDRRFVIKTVSSEDVAEMHNILKKYHQFIVECHGNTLLPQFLGMYRLTVDGVETYMVVTRNVFSHRLTVHRKYDLKGSTVAREASDKEKAKDLPTFKDNDFLNEGQKLHVGEESKKNFLEKLKRDVEFLAQLKIMDYSLLVGIHDVDRAEQEEMEVEERAEDEECENDGVGGNLLCSYGTPPDSPGNLLSFPRFFGPGEFDPSVDVYAMKSHESSPKKEVYFMAIIDILTPYDTKKKAAHAAKTVKHGAGAEISTVNPEQYSKRFNEFMSNILT
  
Inhibitor
Name:
BDBM691393
Synonyms:
US20240277852, Compound 12
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
Search PDB for entries with ligand similarity: