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Target
Sphingosine 1-phosphate receptor 2
Ligand
BDBM31042
Substrate
n/a
Meas. Tech.
Dose Response Cell Based Assay for Antagonists of the S1P2 Receptor
IC50
6211±n/a nM
Citation
 PubChem, PC Dose Response Cell Based Assay for Antagonists of the S1P2 Receptor PubChem Bioassay (2007)[AID] 
Target
Name:
Sphingosine 1-phosphate receptor 2
Synonyms:
EDG5 | S1P2 | S1PR2 | S1PR2_HUMAN | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor Edg-5 | Sphingosine-1-phosphate receptor 2 | ndothelial differentiation G-protein coupled receptor 5
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38883.16
Organism:
Homo sapiens (Human)
Description:
Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay.
Residue:
353
Sequence:
MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVARNSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASVFSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACSTVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLGVFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVLRPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV
  
Inhibitor
Name:
BDBM31042
Synonyms:
(5-acetamido-4-acetyloxy-2,1,3-benzoxadiazol-7-yl) acetate | (5-acetamido-4-acetyloxy-2,1,3-benzoxadiazol-7-yl) ethanoate | Acetic acid 7-acetoxy-5-acetylamino-benzo[1,2,5]oxadiazol-4-yl ester | MLS000077136 | SMR000008576 | acetic acid (5-acetamido-4-acetyloxy-2,1,3-benzoxadiazol-7-yl) ester | acetic acid (6-acetamido-7-acetoxy-benzofurazan-4-yl) ester | cid_597363
Type:
Small organic molecule
Emp. Form.:
C12H11N3O6
Mol. Mass.:
293.2322
SMILES:
CC(=O)Nc1cc(OC(C)=O)c2nonc2c1OC(C)=O
Structure:
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