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Target
X-box-binding protein 1
Ligand
BDBM36923
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
3850±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM36923
Synonyms:
(Z)-3,4-bis(benzenesulfonyl)-2-buten-1-ol | (Z)-3,4-bis(benzenesulfonyl)but-2-en-1-ol | (Z)-3,4-bis(phenylsulfonyl)but-2-en-1-ol | (Z)-3,4-dibesylbut-2-en-1-ol | MLS000080860 | SMR000043655 | cid_5389617
Type:
Small organic molecule
Emp. Form.:
C16H16O5S2
Mol. Mass.:
352.425
SMILES:
OC\C=C(\CS(=O)(=O)c1ccccc1)S(=O)(=O)c1ccccc1
Structure:
Search PDB for entries with ligand similarity: