Reaction Details Report a problem with these data
Target
Cannabinoid receptor 2
Ligand
BDBM50454100
Substrate
n/a
Meas. Tech.
ChEMBL_1752022 (CHEMBL4186782)
Ki
>40000±n/a nM
Citation
 Murineddu, G; Deligia, F; Ragusa, G; García-Toscano, L; Gómez-Cañas, M; Asproni, B; Satta, V; Cichero, E; Pazos, R; Fossa, P; Loriga, G; Fernández-Ruiz, J; Pinna, GA Novel sulfenamides and sulfonamides based on pyridazinone and pyridazine scaffolds as CB Bioorg Med Chem 26:295-307 (2018) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CANNABINOID CB2 | CB-2 | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Human
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM50454100
Synonyms:
CHEMBL4206866
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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